Q9Y463 DYRK1B


Group: CMGC
Family: DYRK
PDB Structure Num: 0
FDA approved drugs from DrugBank: Fostamatinib






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
PGPHHJBZEGSUNE-JYRVWZFOSA-N220100%active
BXNJHAXVSOCGBA-UHFFFAOYSA-N440100%active
PKEDBIGNILOTHW-YWEYNIOJSA-N101100%inactive
CLIWAKTWXZNUAC-UHFFFAOYSA-N110100%active
ZBELDPMWYXDLNY-UHFFFAOYSA-N110100%active
ZPXSIWLYMMFFCE-UHFFFAOYSA-N110100%active
ZQVADOVUSXDTNV-UHFFFAOYSA-N110100%active
QSGKPYRFWJINEH-UHFFFAOYSA-N110100%active
VONVAHFLRYRXSJ-UHFFFAOYSA-N110100%active
HFJRGZBUEXFBMO-UHFFFAOYSA-N110100%active
ZSZSXTFUWZNVBW-UHFFFAOYSA-N110100%active
ZLFXEVGPZWFVCB-UHFFFAOYSA-N110100%active
JMENQRYRZLNDDO-UHFFFAOYSA-N110100%active
OTKQTETZDVGXBV-UHFFFAOYSA-N110100%active
QCJWUXFCDRVWGH-UHFFFAOYSA-N110100%active
MDPBVLVUPMAUIA-UHFFFAOYSA-N110100%active
SCSFTOHNPKDROT-UHFFFAOYSA-N110100%active
GDFYUGGDTISZFA-UHFFFAOYSA-N110100%active
QTRQYFCAAHDIDR-UHFFFAOYSA-N110100%active
WYEVMOFRKALLJA-UHFFFAOYSA-N110100%active
BGXZIBSLBRKDTP-UHFFFAOYSA-N110100%active
BIMZUQRAGIDOLB-UHFFFAOYSA-N110100%active
AVKKQBJQERVCTD-UHFFFAOYSA-N110100%active
KIMRTWGQATWAQF-UHFFFAOYSA-N110100%active
ZGFYGZLBXCHRCV-UHFFFAOYSA-N110100%active
OCVVFPATGNRPNO-UHFFFAOYSA-N110100%active
QISBQDNTYJNGHX-UHFFFAOYSA-N110100%active
NFPDLDFOSLPKHQ-UHFFFAOYSA-N110100%active
ZKGOFDAUIALGLZ-UHFFFAOYSA-N110100%active
KNLSVEADBVICIJ-UHFFFAOYSA-N110100%active
OIUXUISHRLJKGO-UHFFFAOYSA-N101100%inactive
PPALZSWDMRGSQV-UHFFFAOYSA-N110100%active
PHNXNPZJZWLACS-UHFFFAOYSA-N101100%inactive
YCEAZZWLNZYSCL-UHFFFAOYSA-N110100%active
OAUMCWJJYNUCIM-UHFFFAOYSA-N110100%active
JQSJAVBMIMDUFO-UHFFFAOYSA-N101100%inactive
MQJVDVMWBFSFHI-UHFFFAOYSA-N110100%active
RMQRHTAARSAOHF-UHFFFAOYSA-N110100%active
ZYPJRFNOUPSZFL-UHFFFAOYSA-N101100%inactive
OKBNCPDNYVDCTG-UHFFFAOYSA-N110100%active
LZUVHLORMNUQJL-UHFFFAOYSA-N101100%inactive
QLSWEZZOYCDEGC-UHFFFAOYSA-N110100%active
INAVVYMHODCJNF-UHFFFAOYSA-N110100%active
KIUXCHKRJQPHFK-UHFFFAOYSA-N101100%inactive
CKKUHARWBUXFAW-UHFFFAOYSA-N110100%active
AGVJTKJACRWQPP-UHFFFAOYSA-N101100%inactive
FFJGYBJUQCZAAY-UHFFFAOYSA-N110100%active
QDNBLKZVYODRLC-UHFFFAOYSA-N110100%active
DKKAPUBGRWMMGK-UHFFFAOYSA-N101100%inactive
GIQDYWGEMOCDSN-UHFFFAOYSA-N110100%active
DNJISDHVBHLOGY-UHFFFAOYSA-N110100%active
SDSQMAISOKRJPN-UHFFFAOYSA-N110100%active
MRWURALZVKJHPD-UHFFFAOYSA-N110100%active
YBASBPWQGVPOIX-UHFFFAOYSA-N110100%active
FPFBUUBVECCCFK-UHFFFAOYSA-N110100%active
IKEGFWWGERPFMP-UHFFFAOYSA-N101100%inactive
MYHMILRQDXANLR-UHFFFAOYSA-N110100%active
SIVLENRHVVVPKJ-UHFFFAOYSA-N110100%active
FSICBNKCBMOCOY-UHFFFAOYSA-N110100%active
CXOICQRVGSVVHC-UHFFFAOYSA-N110100%active
FOGSRCKIVNMUSS-UHFFFAOYSA-N101100%inactive
FRILKPCZRSAZON-UHFFFAOYSA-N110100%active
CQKBSRPVZZLCJE-UHFFFAOYSA-N110100%active
OWEQZGPRBRSUEF-UHFFFAOYSA-N110100%active
OSGPGSKNNFIBDD-UHFFFAOYSA-N101100%inactive
PCIQNDJCGPAWGK-UHFFFAOYSA-N110100%active
RQFGUPSBOAVFSQ-UHFFFAOYSA-N110100%active
JAJFJEDUYYFVEE-UHFFFAOYSA-N110100%active
UTGHIUITNUXCRZ-UHFFFAOYSA-N110100%active
JHKYWRMDSIQKSV-UHFFFAOYSA-N110100%active
MFXSCAPVWMOBTK-UHFFFAOYSA-N101100%inactive
SYYAIOURHWVANM-UHFFFAOYSA-N101100%inactive
QSWUXXLUPIYCHQ-UHFFFAOYSA-N101100%inactive
UTGHIUITNUXCRZ-LJQANCHMSA-N110100%active
UTGHIUITNUXCRZ-IBGZPJMESA-N101100%inactive
KUFCYNGJQRKYSQ-UHFFFAOYSA-N110100%active
VYFQFYLXCQFLON-UHFFFAOYSA-N101100%inactive
GFSFWVNETAIFJQ-UHFFFAOYSA-N110100%active
LZUJDIWVWSRLRQ-UYRXBGFRSA-N110100%active
ZBYBDKHFLSHGBP-QNGOZBTKSA-N110100%active
COUZVMMRGYONAQ-UHFFFAOYSA-N110100%active
BOSSBLQXHFNQIF-UHFFFAOYSA-N110100%active
ZEMYKTSDVYCVHN-UHFFFAOYSA-N101100%inactive
UPQYLOOUUTWYND-UHFFFAOYSA-N101100%inactive
XRLNWNALNXYYBG-UHFFFAOYSA-N101100%inactive
QOXIXYNVZQZUEZ-UHFFFAOYSA-N101100%inactive
GQIHUCLIFWOITE-UHFFFAOYSA-N110100%active
WRKBHVDIKMUHFE-UHFFFAOYSA-N101100%inactive
QUAHGPDRFLAKAC-UHFFFAOYSA-N110100%active
GGYHYBCBNXKDBY-UHFFFAOYSA-N110100%active
JJWSSJTXQDVFBX-UHFFFAOYSA-N101100%inactive
QKNWFPRGYBXQMF-UHFFFAOYSA-N101100%inactive
JUQUOEZMUSCAFN-UHFFFAOYSA-N110100%active
GQVSWGAIIWEDCW-UHFFFAOYSA-N101100%inactive
CPZBJZDKSIASGT-UHFFFAOYSA-N101100%inactive
BMFODXAZKLMRNP-UHFFFAOYSA-N21150%exclude
MGLSXXJUCASPKK-UHFFFAOYSA-N220100%active
GZCPTOJBBPEFMY-UHFFFAOYSA-N220100%active
OEMURATYWKELKJ-UHFFFAOYSA-N110100%active
FAJUKMUPSMAZEK-UHFFFAOYSA-N110100%active
KSIRCFGDZWDBAM-UHFFFAOYSA-N110100%active
CFPNWWZAVOZYGZ-UHFFFAOYSA-N220100%active
ZYVXTMKTGDARKR-UHFFFAOYSA-N220100%active
MHAJGINRQAEMIM-UHFFFAOYSA-N110100%active
JUSBGYZKUCMHQQ-UHFFFAOYSA-N220100%active
DSAZIMVNBOYSQB-UHFFFAOYSA-N220100%active
FTZQWKAIKYEWPM-UHFFFAOYSA-N110100%active
DUQLWBPQEZFAKS-UHFFFAOYSA-N110100%active
XPBRJXPIAAHIDG-UHFFFAOYSA-N110100%active
QEASAEABBPXQEO-UHFFFAOYSA-N21150%exclude
UTJIEBWCJRJUNS-UHFFFAOYSA-N21150%exclude
WDJPGJTYVFXRTA-UHFFFAOYSA-N21150%exclude
SSUYSUSCBUXMBR-VOTSOKGWSA-N220100%active
VAXXXDBEUYQWBN-UHFFFAOYSA-N21150%exclude
CZCUSHJQJWKYTD-UHFFFAOYSA-N220100%active
OAAPSDVPLURZJC-UHFFFAOYSA-N220100%active
VZGXJTZKPDEJGJ-UHFFFAOYSA-N110100%active
ABRIIMZXUFHPCH-UHFFFAOYSA-N110100%active
PCUWPDUAQBAWHT-UHFFFAOYSA-N110100%active
SDRAETFVRBBLOB-UHFFFAOYSA-N101100%inactive
UWOGNCRXEQLSQQ-UHFFFAOYSA-N101100%inactive
WXMYTQDKBPDSSR-UHFFFAOYSA-N101100%inactive
ARYGGCNDASPYNG-UHFFFAOYSA-N110100%active
WGBRJADREQKUMW-UHFFFAOYSA-N101100%inactive
WYQPGNJIFZHADC-UHFFFAOYSA-N101100%inactive
VCFPJHJKTXRDGD-UHFFFAOYSA-N101100%inactive
MUVCSDSMBYPVGX-UHFFFAOYSA-N101100%inactive
WNKQZLFWZLQFOH-UHFFFAOYSA-N110100%active
MBSKMEQHKIKWQZ-CSKARUKUSA-N101100%inactive
UZLHPXPKYRQXJV-WEVVVXLNSA-N101100%inactive
ZFGAUFCQRUSRCF-XFFZJAGNSA-N110100%active
HGZJFYKLDIBVKD-TWGQIWQCSA-N101100%inactive
AGAPXMAFESZJGN-JXMROGBWSA-N101100%inactive
FMOOGIYSVBVFIT-WEVVVXLNSA-N101100%inactive
TZQCWGJVIDIVCF-PKNBQFBNSA-N101100%inactive
DMARRXYRWLAEFB-POHAHGRESA-N110100%active
WBCONKPHYUGGFA-XYOKQWHBSA-N101100%inactive
JZCVQLIASALOPP-FMIVXFBMSA-N101100%inactive
TWNKLQGDXMYCCB-WTKPLQERSA-N110100%active
MTQKRKLSQROTRY-BJMVGYQFSA-N101100%inactive
KVKWXEDCCDYLBI-BAQGIRSFSA-N101100%inactive
UKFPGYWBGLNLOJ-DHZHZOJOSA-N101100%inactive
ORGCJYCWFZQEFX-RMKNXTFCSA-N101100%inactive
ONYWBNVSVNXDNV-DHZHZOJOSA-N101100%inactive
SQWZFLMPDUSYGV-POHAHGRESA-N110100%active
FBMJGDCKBKUMJF-UHFFFAOYSA-N110100%active
BYUPNMOFJSAIHN-KPKJPENVSA-N110100%active
MHURZKJMJCNXDR-UHFFFAOYSA-N110100%active
TZFBRBFUNGMUNQ-UHFFFAOYSA-N110100%active
PAHHKMMVQJCPJI-UHFFFAOYSA-N110100%active
UVJQEKJPAVSBTA-UHFFFAOYSA-N110100%active
LKROTCXRJRCMTD-UHFFFAOYSA-N110100%active
UFGCTWUIESUHQP-UHFFFAOYSA-N110100%active
NJETXHOGHMMTEB-KPKJPENVSA-N110100%active
GQBQUBULFDQKBM-UHFFFAOYSA-N110100%active
WAJNOEPHTZIWTO-UHFFFAOYSA-N110100%active
SMVHCOBBHAPLPU-UHFFFAOYSA-N101100%inactive
RWAVDFHFFDMSHX-UHFFFAOYSA-N110100%active
JIPWXCWXQYQCQS-UHFFFAOYSA-N101100%inactive
ZNBZVAGNLWMGJD-UHFFFAOYSA-N101100%inactive
RJJPKHZEICLSQD-UHFFFAOYSA-N101100%inactive
UHOPJKMQVDXYAV-UHFFFAOYSA-N110100%active
YPTMZNNBDPEMOK-UHFFFAOYSA-N110100%active
ZDINVWCJHPMIKS-UHFFFAOYSA-N110100%active
FMTZJHHPYOHWNQ-UHFFFAOYSA-N101100%inactive
UUIPRATXTHJYHH-UHFFFAOYSA-N110100%active
GPMRASYSIQENIJ-UHFFFAOYSA-N110100%active
JJUHKRNDDMOYGK-UHFFFAOYSA-N110100%active
WKDIVCXCWMVLPY-UHFFFAOYSA-N110100%active
PVFNDFZQGWYILU-UHFFFAOYSA-N110100%active
BUDHBLBYISRDCR-UHFFFAOYSA-N110100%active
UDBMFFIMVBBFKP-UHFFFAOYSA-N110100%active
XVVPNHZWUXCHJE-UHFFFAOYSA-N110100%active
KOMXYYABYRRJBD-UHFFFAOYSA-N110100%active
ATXGVVQAUKKFAN-UHFFFAOYSA-N110100%active
QZIYOWZOZNSBGJ-UHFFFAOYSA-N110100%active
DPSFKKBIIZTWDA-UHFFFAOYSA-N110100%active
BHKVSOQUPYXVRZ-AWEZNQCLSA-N101100%inactive
HHUOQHKKRABAQB-UHFFFAOYSA-N110100%active
CWJLAVRXVFHDSJ-UHFFFAOYSA-N110100%active
OEQGSMAROCJMFY-UHFFFAOYSA-N101100%inactive
YGXHQYJKJUFSJI-AWEZNQCLSA-N110100%active
RWVARJSWZIIHSJ-JTQLQIEISA-N101100%inactive
CQZSVQKINMHLBO-ZDUSSCGKSA-N110100%active
IVGVIXYZACDUMF-UHFFFAOYSA-N101100%inactive
CEHSVNYYAPNMFI-UHFFFAOYSA-N101100%inactive
FTGAOPZDJRWUTG-FRSZACSASA-N110100%active
DKGZXXQSVKWPRW-NSHDSACASA-N101100%inactive
YJKLTUUIJIUZDP-UHFFFAOYSA-N101100%inactive
FABGVXWXZKTQBP-UHFFFAOYSA-N101100%inactive
RVNDFXJEYCICIV-ZDUSSCGKSA-N110100%active
SZOYOCHRMSEEMG-AIHKSIKWSA-N110100%active
GVANUSPDJMCBIK-UHFFFAOYSA-N101100%inactive
MQUIMJBWAKAKBG-CPMYVITQSA-N101100%inactive
DSCUTYQYWCTFQL-HNNXBMFYSA-N110100%active
KCXBBJNHGRCSQQ-IRXDYDNUSA-N101100%inactive
UTDNMHFLZJFPPY-LZYBPNLTSA-N110100%active
VBYRFFCBZNEHAL-CYBMUJFWSA-N110100%active
AINKQRBPBUTJRM-UHFFFAOYSA-N110100%active
DZYTUBQFYNVYGA-UHFFFAOYSA-N101100%inactive
DPVHKRYDZPCZCT-CYBMUJFWSA-N101100%inactive
WLUFZZMAAGDSJH-UHFFFAOYSA-N101100%inactive
KCXBBJNHGRCSQQ-IAGOWNOFSA-N101100%inactive
FFYSXJWQSSBECR-UHFFFAOYSA-N101100%inactive
XLUOKXQFFGFGNB-UHFFFAOYSA-N101100%inactive
WSUWIXYPBRLNOT-FRKPEAEDSA-N101100%inactive
KCXBBJNHGRCSQQ-SJORKVTESA-N101100%inactive
HTNKXRHQVGPWRO-UHFFFAOYSA-N101100%inactive
WSIMQBVAVXJVGA-UHFFFAOYSA-N101100%inactive
QQCCFMCJVKPTMI-ZDUSSCGKSA-N101100%inactive
FJAIARRQBXWUMX-VIFPVBQESA-N101100%inactive
SZOYOCHRMSEEMG-HFRLZFEPSA-N110100%active
AMUFSGPBIFOSNV-ZDUSSCGKSA-N110100%active
XDTSBZLQROEIPM-UHFFFAOYSA-N101100%inactive
PSHWYQXGQNRHHK-ZDUSSCGKSA-N101100%inactive
QPIYTIVQAQQCFP-UHFFFAOYSA-N101100%inactive
LZRHAZRGHSSHLR-ZDUSSCGKSA-N110100%active
XNYOTZHBHJIMBV-UHFFFAOYSA-N101100%inactive
HMMICWRUNSZYCJ-AWEZNQCLSA-N101100%inactive
GQHOZRVWFHUSGK-UHFFFAOYSA-N101100%inactive
HHTIJHCFCZBRNC-JTQLQIEISA-N101100%inactive
WCXPUTJZKXHALD-ZDUSSCGKSA-N101100%inactive
YELPLVUUDHOICI-KRWDZBQOSA-N110100%active
OHARPIGKJAKOCM-AWEZNQCLSA-N110100%active
DPVHKRYDZPCZCT-ZDUSSCGKSA-N101100%inactive
SOIYEAXWSCNVLD-SNAWJCMRSA-N101100%inactive
OJYINLHOEHUFHI-NSHDSACASA-N110100%active
UIQXQUINYXMORH-UHFFFAOYSA-N101100%inactive
KCXBBJNHGRCSQQ-DLBZAZTESA-N101100%inactive
PDJLHUHTIYCYTA-LBPRGKRZSA-N101100%inactive
WEQRXDXDFLBIDK-UHFFFAOYSA-N110100%active
IZURDRXMCYDUFB-ZDUSSCGKSA-N101100%inactive
KAGWQDFFFLWBFD-ZDUSSCGKSA-N110100%active
QJRRYVISMPFJOU-UHFFFAOYSA-N110100%active
NIVGEZBXSVDFEA-UHFFFAOYSA-N101100%inactive
SEERTRJTWMFXIC-UHFFFAOYSA-N101100%inactive
IOJVCHVCXVTROS-UHFFFAOYSA-N101100%inactive
LKIALHRKZQTCAU-UHFFFAOYSA-N101100%inactive
XKEVCFMQXOOMNO-UHFFFAOYSA-N101100%inactive
XFXMKQIXGVZQIA-UHFFFAOYSA-N101100%inactive
PBNKEANYJCQEQI-KAMYIIQDSA-N101100%inactive
ASDQMECUMYIVBG-UHFFFAOYSA-N101100%inactive
CQNULDWOIXHYFM-SILNSSARSA-N101100%inactive
NNSGCMOBDRALMM-UHFFFAOYSA-N101100%inactive
GZABGNNMQYCDLS-UHFFFAOYSA-N101100%inactive
REHULOMJRMEOTO-UHFFFAOYSA-N101100%inactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N101100%inactive
XLTKBDZXXGQCSC-TWGQIWQCSA-N101100%inactive
DSISPBFCWKLZEA-UHFFFAOYSA-N101100%inactive
MDWXVGCLSBQVMP-UHFFFAOYSA-N101100%inactive
IGRYEDIMNMEBBU-UHFFFAOYSA-N101100%inactive
WHFIWINTCCNYQZ-UHFFFAOYSA-N101100%inactive
BUEJIFZTPCLPMU-UHFFFAOYSA-N101100%inactive
OYTWHNGVDJBJBY-UHFFFAOYSA-N101100%inactive
HJSBIVFFPRFFDM-UHFFFAOYSA-N101100%inactive
FKVVLDSZZBRLMW-UHFFFAOYSA-N101100%inactive
CMLCCTPKLYKIJA-UHFFFAOYSA-N101100%inactive
DRJPJGLJJAOLKO-UHFFFAOYSA-N101100%inactive
DDXAAHDVGNFNMM-UHFFFAOYSA-N101100%inactive
GWGKDCYRVAQDDJ-LFAOLKIESA-N101100%inactive
CEIVAPWZRJLAEW-UHFFFAOYSA-N101100%inactive
RUXUZBIASAPEFP-UHFFFAOYSA-N101100%inactive
JNNGGJDFTJICDZ-AATRIKPKSA-N101100%inactive
ZMXZKIHBCFYBTC-UHFFFAOYSA-N101100%inactive