Q13153 PAK1


Group: STE
Family: STE20
PDB Structure Num: 20
FDA approved drugs from DrugBank: Fostamatinib






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
FTGUWURNNBVUBC-UHFFFAOYSA-N110100%active
PVZRBQHDDWNKDW-ZDUSSCGKSA-N110100%active
GHYZGSZITPRQRZ-UHFFFAOYSA-N110100%active
WTEGSNARHOVIJM-NUHJPDEHSA-N110100%active
ZLZJYPLAARWUEF-UHFFFAOYSA-N110100%active
DBXCSUGFLBSBAW-UHFFFAOYSA-N110100%active
NJAOQMIGMQGBPU-UHFFFAOYSA-N110100%active
JHSXCPVQTSCITM-UHFFFAOYSA-N110100%active
LYPJJBGYRGFAOQ-UHFFFAOYSA-N110100%active
JDOMJOMBOYZLKG-UHFFFAOYSA-N101100%inactive
WTANZLLBRSOYBE-UHFFFAOYSA-N101100%inactive
ANMMEXVLDZGIOZ-UHFFFAOYSA-N101100%inactive
BNOUWVFOOUWOLD-UHFFFAOYSA-N101100%inactive
LCGPOGPEUQTXLK-UHFFFAOYSA-N101100%inactive
HJDWTGMIRQXKFE-UHFFFAOYSA-N101100%inactive
WNJHVJCQNWZLPX-UHFFFAOYSA-N101100%inactive
RAOHJDZUEDDWGV-UHFFFAOYSA-N101100%inactive
KCKDYWFERPXFNA-UHFFFAOYSA-N101100%inactive
XQKDYHDILSOXNK-UHFFFAOYSA-N101100%inactive
MRYXWSRMKBRWDF-UHFFFAOYSA-N110100%active
JTSOHDVEOQCKQO-UHFFFAOYSA-N101100%inactive
ODDOXBDADZOQGE-UHFFFAOYSA-N101100%inactive
MEOWYSKGQKBNMJ-UHFFFAOYSA-N101100%inactive
QSXRGEQOCHJNOT-UHFFFAOYSA-N101100%inactive
VXKHKPJWTVBJQO-UHFFFAOYSA-N101100%inactive
LYGWGCZJFVDMES-UHFFFAOYSA-N101100%inactive
VITDSSKYLOCDAP-UHFFFAOYSA-N110100%active
AHQWIBJDMASYON-UHFFFAOYSA-N110100%active
AHQWIBJDMASYON-KRWDZBQOSA-N110100%active
AHQWIBJDMASYON-QGZVFWFLSA-N110100%active
RZXMIHOUHYSGJO-UHFFFAOYSA-N202100%inactive
NDZPPXQOOUNQTQ-UHFFFAOYSA-N101100%inactive
TUBDCTXNBUJRCI-AULYBMBSSA-N101100%inactive
SGUZXWKWTMWMCR-LBPRGKRZSA-N110100%active
DXUVJKCCXSAUKZ-NSHDSACASA-N110100%active
DYLHVDVCWIEYSA-UHFFFAOYSA-N110100%active
LDWBULFGVRAVMR-UHFFFAOYSA-N110100%active
LXAVLHJMLKIDME-UHFFFAOYSA-N110100%active
CYXJGDDHTZEOTA-CYBMUJFWSA-N101100%inactive
ZGYNHFQKPDQJBV-UHFFFAOYSA-N110100%active
UIBDEIGYCMBVOR-UHFFFAOYSA-N21150%exclude
FPENQVXQIUJGIO-UHFFFAOYSA-N110100%active
RBILTCANHJYJDG-UHFFFAOYSA-N101100%inactive
KQGMUUYYFGZQDW-UHFFFAOYSA-N110100%active
CYBQVRXXIUXCHG-UHFFFAOYSA-N110100%active
AVBHAEAKXMFDFJ-UHFFFAOYSA-N110100%active
XTBHQOFIMLVUIZ-UHFFFAOYSA-N101100%inactive
JWIKJMNJZBWYTQ-UHFFFAOYSA-N110100%active
WQKUSPIXIQAONS-UHFFFAOYSA-N101100%inactive
AJHFOGJCDKOZKC-UHFFFAOYSA-N110100%active
WJRJVWODJIJPTO-UHFFFAOYSA-N101100%inactive
AHCUZFSXUJVVCW-UHFFFAOYSA-N110100%active
NFQOHAZHLGREAU-UHFFFAOYSA-N110100%active
RHZPBNHUNKAZOC-UHFFFAOYSA-N110100%active
RHUNVKDQHRRINU-UHFFFAOYSA-N101100%inactive
AQSFORPPQYDEMZ-UHFFFAOYSA-N110100%active
XPRBQHYGBQLJPC-UHFFFAOYSA-N110100%active
ZVLBZKCPVGAIDV-UHFFFAOYSA-N110100%active
ZRLGRLKEULDQNW-UHFFFAOYSA-N101100%inactive
IJWZHPQMDARGAM-UHFFFAOYSA-N110100%active
RTPZFHYRWPLORR-UHFFFAOYSA-N110100%active
ZERPGXMMUNAELZ-UHFFFAOYSA-N110100%active
KYIWCGBICYODPB-UHFFFAOYSA-N110100%active
RNUSQJPABDFZQP-UHFFFAOYSA-N110100%active
ZTABOYRFNXBMEJ-UHFFFAOYSA-N110100%active
RYCCEJFMPINKHD-UHFFFAOYSA-N110100%active
PLVWOAJTKKTTSU-UHFFFAOYSA-N110100%active
SZEDQVIUDYYZDB-UHFFFAOYSA-N110100%active
DLPXGJYWIQSIOJ-UHFFFAOYSA-N110100%active
HVSVERGUSJAVSI-UHFFFAOYSA-N110100%active
JBKAGOBFGDHBNE-UHFFFAOYSA-N110100%active
YNRKCDBURYJRQF-UHFFFAOYSA-N110100%active
GYOYJIDGMCNEHB-UHFFFAOYSA-N21150%exclude
GTSQIGNGTWZBMV-UHFFFAOYSA-N21150%exclude
UOQSDEILBQECQK-UHFFFAOYSA-N220100%active
CSZDODQDQINNHM-UHFFFAOYSA-N21150%exclude
NDESJLVJOXCZGF-UHFFFAOYSA-N220100%active
PYSIAKZWZJNMNM-UHFFFAOYSA-N202100%inactive
DGBFDSJYMVTWOH-UHFFFAOYSA-N505100%inactive
NQBRFDSRSGHBBK-UHFFFAOYSA-N110100%active
GKEGWJJRPYLMOW-KRWDZBQOSA-N110100%active
NIVBGOGCJSMNMG-KRWDZBQOSA-N110100%active
OINGHOPGNMYCAB-INIZCTEOSA-N110100%active
AYCPARAPKDAOEN-LJQANCHMSA-N220100%active
DHUJCQOUWQMVCG-UHFFFAOYSA-N330100%active
DHKFOIHIUYFSOF-UHFFFAOYSA-N110100%active
RFAXLXKIAKIUDT-UHFFFAOYSA-N101100%inactive
HWHNITBPQIFDQC-RUCARUNLSA-N110100%active
SGTPEULULIFDRG-RXAXNXDRSA-N110100%active
ZVGQZSQDTLALCO-SFHVURJKSA-N110100%active
GMQHFTHVKUIAEO-UHFFFAOYSA-N110100%active
GYMFXAFMBGPIFA-UHFFFAOYSA-N101100%inactive
RYCBSFIKWACFBY-UHFFFAOYSA-N110100%active
MIKSFVUBHJVZMS-VVOJOOEHSA-N110100%active
UFUJWBLMFIYWJW-UHFFFAOYSA-N110100%active
QEFLWXKYNFVJSP-UHFFFAOYSA-N110100%active
ZBCMHWUFWQFPLV-VVOJOOEHSA-N110100%active
PKIRBWTZDHRUJE-XGAFWQRZSA-N110100%active
ICNMDSYSAGMRJC-UHFFFAOYSA-N101100%inactive
PJYRMGKJLXENCU-IRJFHVNHSA-N110100%active
BSGQVUPHCVNSRM-QGZVFWFLSA-N110100%active
GUERACYCGKAFOU-LLVKDONJSA-N101100%inactive
IVWHSTCJCURGMH-UHFFFAOYSA-N21150%exclude
QSTNFLZQNNYKIM-UHFFFAOYSA-N220100%active
VWEBEVMRPSIULB-UHFFFAOYSA-N21150%exclude
YFAWTHFQZWOEJN-UHFFFAOYSA-N220100%active
BKHJHXMKWIXRTE-UHFFFAOYSA-N220100%active
ZMBVLMGGQSTPCK-UHFFFAOYSA-N220100%active
WPFLVPJXKWCRQK-UHFFFAOYSA-N330100%active
VPSBNPIVVHGVAY-UHFFFAOYSA-N32166.67%exclude
IPKFWIAZRFRRRB-UHFFFAOYSA-N220100%active
MUTUMOBIBVSADG-UHFFFAOYSA-N21150%exclude
WUHYQOAIEQUWNC-UHFFFAOYSA-N21150%exclude
JYNFBQCZUVMNJC-UHFFFAOYSA-N220100%active
CPBPBGYLBWTBJR-UHFFFAOYSA-N21150%exclude
XHLWSDNRXILCDY-UHFFFAOYSA-N21150%exclude
PNRMHHJAFUYMEV-VXKWHMMOSA-N220100%active
BCGFTSYNPJUGDC-UHFFFAOYSA-N21150%exclude
AHRSJDAOQNYYAI-UHFFFAOYSA-N220100%active
XLFNLJYGUOLEJS-SFHVURJKSA-N101100%inactive
AFLUUMVQPAIWBM-UHFFFAOYSA-N110100%active
OZWKMVRBQXNZKK-UHFFFAOYSA-N101100%inactive
UJYHOKCIZXHJLJ-UHFFFAOYSA-N110100%active
NZCHGHMPHKCWLR-UHFFFAOYSA-N101100%inactive
RXPZOSHFGJWSLQ-UHFFFAOYSA-N101100%inactive
XPWVBCAWYZGUPL-HXUWFJFHSA-N101100%inactive
SCTRERISNHFYGN-LJQANCHMSA-N101100%inactive
BNRXMSGHPVYSDK-UHFFFAOYSA-N101100%inactive
ZDSMRCALKWRRFK-RBSFLKMASA-N101100%inactive
XQFLBDFFGHEFGF-BZUAXINKSA-N101100%inactive
VBYMFAOTZHNONG-UHFFFAOYSA-N101100%inactive
WAAWETUDFSIYSD-UHFFFAOYSA-N101100%inactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N101100%inactive