Q12866 MER


Group: TK
Family: Axl
PDB Structure Num: 12
FDA approved drugs from DrugBank: Fostamatinib






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
JGEBLDKNWBUGRZ-HXUWFJFHSA-N110100%active
OGEBRHQLRGFBNV-RZDIXWSQSA-N220100%active
BQICBFKSXAVIBF-UHFFFAOYSA-N110100%active
ZXZLVQGNVOKCAS-UHFFFAOYSA-N101100%inactive
VDKBGBCLPKTOGS-UHFFFAOYSA-N101100%inactive
XYASHXPUZJDWIO-UHFFFAOYSA-N101100%inactive
NPVXOWLPOFYACO-XUTJKUGGSA-N220100%active
FWSIMUXTYLCNLB-UAPYVXQJSA-N110100%active
HSKPWLBWANOLQJ-XUTJKUGGSA-N110100%active
JMWVQYVMGWIDOO-XUTJKUGGSA-N110100%active
WHWWZWPSOQJMQR-UAPYVXQJSA-N110100%active
KSWWEWKERJBYBF-UAPYVXQJSA-N110100%active
RIDPOYWCOSZKLX-UAPYVXQJSA-N110100%active
NVGYLVRTAGAASJ-AQYVVDRMSA-N110100%active
QEGOHWRXPWNJLM-XGAFWQRZSA-N110100%active
KNJWVKYCJCNLTC-AFARHQOCSA-N110100%active
IJBQYPBBOUFSEN-WGSAOQKQSA-N110100%active
ZQOUBHKEPWWNKQ-UHFFFAOYSA-N101100%inactive
CSTHTXUPJYUFSY-UHFFFAOYSA-N110100%active
JGSVNIPAOGOWTI-LJQANCHMSA-N110100%active
GSYCGAZRNZUCGI-UHFFFAOYSA-N110100%active
PUVADVGBMMQLRI-GOSISDBHSA-N101100%inactive
PUVADVGBMMQLRI-SFHVURJKSA-N110100%active
IFGAKKDJKVVCHX-UHFFFAOYSA-N101100%inactive
PGCRMYCYVMGKSR-UHFFFAOYSA-N110100%active
HYJQBVXSXMOCKZ-UHFFFAOYSA-N101100%inactive
NQSZPRKIVXBBNI-KOMQPUFPSA-N101100%inactive
XCVFEECOCBFREB-JCNLHEQBSA-N110100%active
WCBFHMOPYCFZQV-SAABIXHNSA-N110100%active
DKLRVMHGCQHXBG-UAPYVXQJSA-N110100%active
CVMMQZHPZPFORW-KOMQPUFPSA-N110100%active
SYMFPMGEVCPXSZ-QAQDUYKDSA-N110100%active
FDBSFRHJILHTNZ-JCNLHEQBSA-N110100%active
VDZKYCXBCMIQDA-JCNLHEQBSA-N110100%active
AXMGRXURKXGCPI-JCNLHEQBSA-N110100%active
OPZZIKZUGSMEPY-WKILWMFISA-N110100%active
MNAFIBDUOJAZPP-XGAFWQRZSA-N110100%active
FJWZASZEWLWFRB-AQYVVDRMSA-N110100%active
DKAWAHOTJBIOOP-KESTWPANSA-N110100%active
DERKWJPZXYTPTQ-IYARVYRRSA-N110100%active
CQFHCAGCNILQLR-QAQDUYKDSA-N110100%active
DLNOLRVJSOGNNN-JCNLHEQBSA-N110100%active
VAWPQSJYRPQHIP-SHTZXODSSA-N110100%active
XUYGOTAWDBTFJQ-WKILWMFISA-N101100%inactive
ZSOMRVGPVJNHFO-KOMQPUFPSA-N110100%active
SOXQFVHZJHSFSW-WKILWMFISA-N101100%inactive
CXDXWPGEWIRDBS-UAPYVXQJSA-N110100%active
WRYYRMHEPCBQIZ-JCNLHEQBSA-N110100%active
IQJYTBNFPSQTDY-RZDIXWSQSA-N101100%inactive
HSYSSKFCQHXOBP-MXVIHJGJSA-N220100%active
HVIDXJFXDHKCMO-UHFFFAOYSA-N110100%active
PUNWZJKAQIQKQL-ZIAGYGMSSA-N110100%active
ZUKWHYJJSUVIEH-JOCQHMNTSA-N110100%active
BQWLIDAUTKRGNB-UHFFFAOYSA-N101100%inactive
KKAICBOHJLVDCE-UHFFFAOYSA-N101100%inactive
KUEUDYJDIPJMFW-HAQNSBGRSA-N101100%inactive
JUUYWFQCWXBEPH-HAQNSBGRSA-N101100%inactive
VMVCKKNFEIDAEX-JOCQHMNTSA-N110100%active
IPLZGPIOLOENJW-HDJSIYSDSA-N110100%active
DBWBCGYTGWUQRF-WKILWMFISA-N110100%active
GJZCXJLZZFATOM-KURUOMIPSA-N110100%active
NZKWELHADKRVPQ-WKILWMFISA-N110100%active
BXVCQFJVWUUMKU-WKILWMFISA-N101100%inactive
YYCBPQHVOAJHLZ-QAQDUYKDSA-N110100%active
OVPGPUIOPKYMQR-IYARVYRRSA-N110100%active
MXSXJVUUCUTMAN-WGSAOQKQSA-N110100%active
CTKKZYMHCDCJTB-JOCQHMNTSA-N110100%active
ISCXJKAZTPOPNW-HDJSIYSDSA-N110100%active
RTLVYUQCERXOJO-SHTZXODSSA-N110100%active
DMDQOCLVSGUEJT-SHTZXODSSA-N110100%active
QFFRGXIFYGLMLF-WKILWMFISA-N101100%inactive
WORRXRIVSMTSEB-WKILWMFISA-N110100%active
QBCMBQCPRNSFJE-MXVIHJGJSA-N110100%active
ZTFAJUAGQGVBCO-KESTWPANSA-N110100%active
NEZRLVDPFUFEKB-MXVIHJGJSA-N110100%active
WQLWLOMHWYQNFN-IYARVYRRSA-N110100%active
XEHHSTXCXVSYIR-IYARVYRRSA-N110100%active
WZSUDZDKYJWJPS-XUTJKUGGSA-N110100%active
BONBXBPLENOTTM-XUTJKUGGSA-N110100%active
WERQRDFKILOXSK-HZCBDIJESA-N110100%active
PWOIRDUWFWWFMT-WGSAOQKQSA-N110100%active
NLXWFBBYANWXPR-IYARVYRRSA-N110100%active
CURNCKHFJSIYBK-UHFFFAOYSA-N101100%inactive
JNYMZWUOQWXOII-SHTZXODSSA-N110100%active
AGYRCBTVZCTMOP-WKILWMFISA-N110100%active
OIVLGMGZZCFPCM-UHFFFAOYSA-N110100%active
OYQORZDLJYKSEI-QAQDUYKDSA-N101100%inactive
TWOVQCHDPBWOKT-HAQNSBGRSA-N101100%inactive
HTOALBYXWRQRAR-SHTZXODSSA-N110100%active
YVAPXKWBCBCTDS-KESTWPANSA-N110100%active
XYSYRHAUHUPOHK-MEMLXQNLSA-N110100%active
ARSCEEUSPNVXQA-UHFFFAOYSA-N110100%active
KAAPXWSYROPAEL-MXVIHJGJSA-N220100%active
DCFNMFYAKVXCLN-MEMLXQNLSA-N110100%active
LFOWPAZJQIZNHI-MEMLXQNLSA-N110100%active
MJSHVHLADKXCML-RQNOJGIXSA-N330100%active
LBEJYFVJIPQSNX-SOAUALDESA-N110100%active
OXQTXNVWTNDAQF-UHFFFAOYSA-N101100%inactive
UQKLTKAHTNLXPA-JOCHJYFZSA-N101100%inactive
QSGGLLCPVRJDDE-JOCHJYFZSA-N101100%inactive
HMMJKDJDJCYCBK-UHFFFAOYSA-N101100%inactive
QXDLEVGKYBDDKC-UHFFFAOYSA-N101100%inactive
AFNWKIKMTQIWHU-UHFFFAOYSA-N101100%inactive
PXQXFGCRWHTVBD-UHFFFAOYSA-N101100%inactive
IJLDJEASLDJCDS-UHFFFAOYSA-N101100%inactive
MJCJKFFVCHBTSF-UHFFFAOYSA-N101100%inactive
QDFNTPGVPJPEHU-UHFFFAOYSA-N101100%inactive
NKKKHNIEVNYMCR-UHFFFAOYSA-N101100%inactive
HKIFQJOVGYXXBB-UHFFFAOYSA-N101100%inactive
RQKOQBFNLXPPSW-UHFFFAOYSA-N101100%inactive
RMRSKURFSGCSFM-UHFFFAOYSA-N101100%inactive
ZEXOTOJJEIBRDN-UHFFFAOYSA-N101100%inactive
FHJDQALLIXLBIE-UHFFFAOYSA-N101100%inactive
XMKZPZBUKQMHNF-UHFFFAOYSA-N101100%inactive
RANDQPGUBTWPSC-UHFFFAOYSA-N101100%inactive
QGEAHLONJRLMKZ-UHFFFAOYSA-N101100%inactive
RCINICONZNJXQF-MZXODVADSA-N101100%inactive
BPOGHKOSOWZBGZ-MHZLTWQESA-N110100%active
NGJAXUZGEAUCFH-UHFFFAOYSA-N110100%active
GUZDWCGVMFWILW-UHFFFAOYSA-N110100%active
TUSFBIZKPNHLKT-UHFFFAOYSA-N110100%active
LZPFBEBTZBKKFB-UHFFFAOYSA-N110100%active
RADSRRYRWZKEEW-UHFFFAOYSA-N110100%active
SDWTWVXMBPUQSC-UHFFFAOYSA-N110100%active
YXLDQBFWFZDCOF-UHFFFAOYSA-N110100%active
RSCAIJXVGDMQRL-UHFFFAOYSA-N110100%active
XBFYWJOKBDZTSR-UHFFFAOYSA-N110100%active
LZOJVTCTBSNNNT-UHFFFAOYSA-N110100%active
XXEJLOWSXIMQHG-UHFFFAOYSA-N110100%active
VNERMGVCIRNEMM-SANMLTNESA-N110100%active
JJXRAZVLEQHSOL-UHFFFAOYSA-N110100%active
ILONTPDVQVKFCL-UHFFFAOYSA-N110100%active
FXTJCTYAPOCFAC-UHFFFAOYSA-N110100%active
BFLSJYFITVZAPW-UHFFFAOYSA-N110100%active
DTHWSLYDAOOPOE-UHFFFAOYSA-N110100%active
SMIXLVLRWCBPBA-UHFFFAOYSA-N110100%active
ZJTWKNHQHNLTPO-UHFFFAOYSA-N110100%active
VPDVHIDCAMWQER-UHFFFAOYSA-N110100%active
UENPHVZMJZONSS-VWLOTQADSA-N110100%active
ORJFNGOUYHBFPE-UHFFFAOYSA-N110100%active
MGGQNMHOSQIZOZ-NDEPHWFRSA-N110100%active
SCCZGJNJWOJDLN-UHFFFAOYSA-N110100%active
DKZQQJXYLNUWFT-LJAQVGFWSA-N110100%active
IKQPJOFHAZFMNC-UHFFFAOYSA-N110100%active
UYSWRVPXWRGZTG-UHFFFAOYSA-N110100%active
UVBALELUPGCHKQ-DEOSSOPVSA-N110100%active
ASMYWCGHYWQPGO-UHFFFAOYSA-N110100%active
GKTJDVXAUIHAML-UHFFFAOYSA-N110100%active
SCPFYDCGZSWLOY-UHFFFAOYSA-N110100%active
CMXOTBPJJMRQOJ-UHFFFAOYSA-N110100%active
SMJAMOAYGIVKRI-UHFFFAOYSA-N101100%inactive
NWXGFDVFXJMUDD-UHFFFAOYSA-N101100%inactive
QXIOZIFTPMAING-VWLOTQADSA-N110100%active
UMBIRSZUCJNBHB-SANMLTNESA-N110100%active
ROHJEIACUNTGFP-VWLOTQADSA-N110100%active
GCDSDVNITVBCDW-VWLOTQADSA-N110100%active
BWCCBKUPFRNBAM-LBPRGKRZSA-N101100%inactive
LNFBAYSBVQBKFR-UHFFFAOYSA-N101100%inactive
YRZPEINIRHVBPS-KESTWPANSA-N101100%inactive
KLCLEAVDENJUGH-SAABIXHNSA-N101100%inactive
WVXVTVISFJYJCL-QAQDUYKDSA-N101100%inactive
RTCOZPJVISFGRP-UHFFFAOYSA-N101100%inactive
FKDZRIQJGKWTDB-MXVIHJGJSA-N101100%inactive
BDVGHJLTQZVVPA-UHFFFAOYSA-N101100%inactive
HLMASOKCFIFSOF-UHFFFAOYSA-N101100%inactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N101100%inactive
YFPYQMFBXQUNHH-UHFFFAOYSA-N101100%inactive
XQEJWZGYFBXKIF-UHFFFAOYSA-N101100%inactive
KXMZDGSRSGHMMK-VWLOTQADSA-N101100%inactive
NRYHKDJEPGDAGX-UHFFFAOYSA-N101100%inactive
ZVIBISIIUYWHAM-UHFFFAOYSA-N101100%inactive
HUZKIRAWCBJPAF-UHFFFAOYSA-N101100%inactive
WXYDWXCNFYMYCG-UHFFFAOYSA-N101100%inactive
PEBCBFJYPZBCNX-UHFFFAOYSA-N101100%inactive
STNFPRBCLKSHGJ-UHFFFAOYSA-N101100%inactive
IWPFYKIFKHNHAS-UHFFFAOYSA-N101100%inactive