Q08881 ITK


Group: TK
Family: Tec
PDB Structure Num: 35
FDA approved drugs from DrugBank: Fostamatinib Pazopanib






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
QAFHWLBRECIPAC-UHFFFAOYSA-N110100%active
ILVXQPRFMVXZRH-UHFFFAOYSA-N101100%inactive
UPBLLWLBMPEKKB-UHFFFAOYSA-N220100%active
IWXOBLGVEGPHBJ-UHFFFAOYSA-N110100%active
MGKBRQHUVOICMA-UHFFFAOYSA-N101100%inactive
PUQHWQFKZDOVQP-UHFFFAOYSA-N101100%inactive
DUXYZTPLTJYCNJ-UHFFFAOYSA-N110100%active
FZABWTFNUIVAHO-UHFFFAOYSA-N110100%active
UBOPXWHTIVENRV-UHFFFAOYSA-N110100%active
WPELVGOARBYVTB-UHFFFAOYSA-N101100%inactive
FUUMUCYFYLYLQL-UHFFFAOYSA-N110100%active
UGLKWJMRDXWSJB-UHFFFAOYSA-N101100%inactive
DQTBORZYKZITIA-UHFFFAOYSA-N110100%active
RWMHHWHCWTVGOV-UHFFFAOYSA-N101100%inactive
UEAQQAPWVJTBSU-UHFFFAOYSA-N110100%active
OZHGDLXRBXUSOS-UHFFFAOYSA-N110100%active
OWIJSXBEEDGYSD-UHFFFAOYSA-N101100%inactive
PKFGOSVXYYLDNY-UHFFFAOYSA-N110100%active
JEGQJSKRWOBVEP-UHFFFAOYSA-N101100%inactive
ZHVDERXJUYELSZ-UHFFFAOYSA-N110100%active
RSJYLNUFSUIOQE-UHFFFAOYSA-N110100%active
PKTNBTZGPAUVEF-UHFFFAOYSA-N110100%active
KARRXYMCFAILBZ-UHFFFAOYSA-N110100%active
QJFLIPZTKYALQR-UHFFFAOYSA-N110100%active
NWUSHDACDTZXCD-UHFFFAOYSA-N101100%inactive
JHBYRHQSNOLZKK-UHFFFAOYSA-N21150%exclude
DWICUERZWRWRJK-UHFFFAOYSA-N101100%inactive
XVZYMHZUVJKMBG-UHFFFAOYSA-N101100%inactive
CFHJARLUPRYYAH-UHFFFAOYSA-N101100%inactive
AFVDQRKAOQLYKF-UHFFFAOYSA-N110100%active
MMBNQDYIJPDYEP-UHFFFAOYSA-N101100%inactive
UCVYWHCLSDDWHR-UHFFFAOYSA-N110100%active
CKYQXIVHGUEYDB-UHFFFAOYSA-N110100%active
NEWALRCVHVFLBK-UHFFFAOYSA-N101100%inactive
FKSIZOYGWLPYOT-UHFFFAOYSA-N101100%inactive
GLJLGEAWRQBSGD-HSZRJFAPSA-N220100%active
CGJVMKJGKFEHTL-HSZRJFAPSA-N220100%active
SJJNZHHGZMUFIM-XMMPIXPASA-N202100%inactive
GLJLGEAWRQBSGD-QHCPKHFHSA-N202100%inactive
MMTIMKJVYCMIOF-HSZRJFAPSA-N110100%active
RMAUIYTVKFMOGP-UHFFFAOYSA-N101100%inactive
PGABPPHMLFSKKA-RTWAWAEBSA-N101100%inactive
WIUYFJQWJMBTCE-UHFFFAOYSA-N110100%active
WIUYFJQWJMBTCE-MOPGFXCFSA-N110100%active
USVGUZMPKPIFFV-MOPGFXCFSA-N101100%inactive
AKDCUCWSQMYOMD-RTWAWAEBSA-N110100%active
QOSKBOUKENYWAA-UHFFFAOYSA-N101100%inactive
LBYBJJIMARLHMV-UHFFFAOYSA-N220100%active
NCXHAHGMYXETMO-QHCPKHFHSA-N220100%active
ZUXTTXJNSUUIGO-JOCHJYFZSA-N110100%active
IGXJXMLDIIGDNE-UHFFFAOYSA-N110100%active
NRJLSFKZAQFLCT-UHFFFAOYSA-N202100%inactive
DTMLASFEUYRUGI-UHFFFAOYSA-N101100%inactive
CMSVKLVKNBMOSI-UHFFFAOYSA-N202100%inactive
STCNDRXGYAQSKS-UHFFFAOYSA-N101100%inactive
SXIQTGHCRRJBCG-UHFFFAOYSA-N101100%inactive
SPABBLGEKOWLOG-UHFFFAOYSA-N101100%inactive
CZAHTSYZRWGJOH-UHFFFAOYSA-N220100%active
COBZZNVRTKQJFM-FQEVSTJZSA-N110100%active
XFYUTGIEFKGWND-NRFANRHFSA-N220100%active
XFYUTGIEFKGWND-OAQYLSRUSA-N101100%inactive
ILYQIAVPXLQYSF-HSZRJFAPSA-N101100%inactive
GLURFGLYQHSJCV-FQEVSTJZSA-N220100%active
IXJCBGOCROYMTK-QFIPXVFZSA-N110100%active
PGNRWZCKDIYZQF-NRFANRHFSA-N110100%active
XHVGFIQVBRHURI-WMZOPIPTSA-N110100%active
GQHAHPQLCBBLDS-IVAFLUGOSA-N220100%active
VQAXOIUGIWGEFE-WBPHRXDCSA-N220100%active
LLHYIISPPGQGTN-JFGZAKSSSA-N220100%active
YXHJHTILTPQTEF-HSZRJFAPSA-N110100%active
TVHDLBOMEGOWNE-SINBQTRASA-N220100%active
SFNLOYSFTSUDRG-IBGZPJMESA-N110100%active
KWTDVQYZRZTJDG-UHFFFAOYSA-N110100%active
SDZFNFGEAWBFTM-DVKBMCPXSA-N110100%active
JNRFIKALOWSUBG-DAVFGYKESA-N110100%active
PTHVKCSYXICMAR-UHFFFAOYSA-N110100%active
UGXCBYVBIJACEK-UHFFFAOYSA-N101100%inactive
SDVAHCXGDGYWFA-UHFFFAOYSA-N110100%active
UMBDWDIRLTVPBF-UHFFFAOYSA-N110100%active
YPXWUKLQAUBCPF-UHFFFAOYSA-N110100%active
ZRYMMWAJAFUANM-INIZCTEOSA-N220100%active
XLFNLJYGUOLEJS-SFHVURJKSA-N101100%inactive
CBRJPFGIXUFMTM-WDEREUQCSA-N101100%inactive
SMJAMOAYGIVKRI-UHFFFAOYSA-N101100%inactive
IOJLBZJSULGZLY-CHHVJCJISA-N101100%inactive
RGNXWPVNPFAADO-NSIKDUERSA-N101100%inactive
OSAWFUCUZJNEID-CQSZACIVSA-N101100%inactive
HDWPLUHUCHVGAN-UHFFFAOYSA-N110100%active
MNFPBGLVKDAKDC-UHFFFAOYSA-N101100%inactive
JUNHKGHGMUGSOV-SNAWJCMRSA-N101100%inactive
CIDLDKKAAKXBML-UHFFFAOYSA-N101100%inactive
GASMTHLXWMOHFL-KPKJPENVSA-N101100%inactive
HEWAPJQDQSFDKB-UHFFFAOYSA-N101100%inactive
IWTXHSVJZHCEOG-UHFFFAOYSA-N101100%inactive
GKTSCCHUGCUTEG-UHFFFAOYSA-N101100%inactive
KESQOYFKTYOFSC-UHFFFAOYSA-N101100%inactive
ZIVOQVDAIKLHOH-UHFFFAOYSA-N101100%inactive
RVSKMYIRDKWVJE-UHFFFAOYSA-N101100%inactive
WYHVICNLFLFZLO-UHFFFAOYSA-N110100%active
VLQPHCSSQQRKAF-UHFFFAOYSA-N101100%inactive
YLDHRDIOVUTLTI-UHFFFAOYSA-N202100%inactive
JRONIANGPGCJCI-UHFFFAOYSA-N101100%inactive
JQOCXCNIIWTKMQ-UHFFFAOYSA-N101100%inactive
XDUXEVVHZJCQJY-UHFFFAOYSA-N101100%inactive
PFFUHUKZADCSFP-UHFFFAOYSA-N110100%active
MCOTWBOPJHLZIX-UHFFFAOYSA-N110100%active
IPSSGRBTYPDFKK-UHFFFAOYSA-N101100%inactive
YOJWQVWRBNADJO-UHFFFAOYSA-N110100%active
VWZPFUCWXLUAGS-UHFFFAOYSA-N101100%inactive
YCQUGZCSTKDMCE-UHFFFAOYSA-N101100%inactive
QGACHVMLSDBCDF-UHFFFAOYSA-N110100%active
YBPAGGHUVVECGN-UHFFFAOYSA-N101100%inactive
CCUMEZRCMJRYHN-UHFFFAOYSA-N101100%inactive
ZSTREMQKBCZVGE-UHFFFAOYSA-N101100%inactive
QTCWXZNSCOYHQN-UHFFFAOYSA-N110100%active
FZWLAIJGXFHQJK-UHFFFAOYSA-N110100%active
DQPJVNQWPBLBAB-UHFFFAOYSA-N220100%active
SRTIAXHDTNPJGI-UHFFFAOYSA-N110100%active
TVEYRZYFTCQNQK-UHFFFAOYSA-N101100%inactive
NEZKYAFRLQAQTL-UHFFFAOYSA-N110100%active
USEKBDKLERFLKV-UHFFFAOYSA-N101100%inactive
NTVGAZWYHVYTIK-UHFFFAOYSA-N101100%inactive
CAMJEDZKEXZNEY-UHFFFAOYSA-N101100%inactive
VTEDTZHIHRZSDP-UHFFFAOYSA-N110100%active
DPCITOXJVNGDHY-UHFFFAOYSA-N101100%inactive
GRBPCANVVVAEQY-UHFFFAOYSA-N110100%active
UWSAYPXXZRHDTN-UHFFFAOYSA-N110100%active
AAFLHABTMIJIEE-UHFFFAOYSA-N110100%active
GKBXPMCATFNHQZ-UHFFFAOYSA-N110100%active
MBQXWTBSEOBPNA-UHFFFAOYSA-N110100%active
VRFYHMPLFWXUSJ-UHFFFAOYSA-N101100%inactive
ZHXNIYGJAOPMSO-UHFFFAOYSA-N110100%active
PGZNWXOKFGIDJL-UHFFFAOYSA-N110100%active
NSUWPDMYMLHMAE-UHFFFAOYSA-N110100%active
KBIXYYWXSZPVEV-UHFFFAOYSA-N110100%active
MCNYWWZQBPAKSM-UHFFFAOYSA-N101100%inactive
CLFOIXVUUDBDGI-UHFFFAOYSA-N110100%active
WPPDGWMXKWIRFC-UHFFFAOYSA-N110100%active
MBSUFDFTBSAUCT-UHFFFAOYSA-N110100%active
YWVLIRJSHTUKIM-UHFFFAOYSA-N110100%active
LYNUPGSZUIJXNJ-UHFFFAOYSA-N101100%inactive
HJANPQFKWPVSDK-UHFFFAOYSA-N101100%inactive
ICLTWMGTAQDABY-UHFFFAOYSA-N110100%active
ZKHQLWLCSPCQIW-UHFFFAOYSA-N101100%inactive
OQNIMKVDOJIQID-UHFFFAOYSA-N110100%active
XIABTCSDBYIJTG-UHFFFAOYSA-N101100%inactive
AUKRLJSUNHCDDH-UHFFFAOYSA-N110100%active
NQJICWCKADTPEW-UHFFFAOYSA-N110100%active
CYENRWZQGSRRDN-UHFFFAOYSA-N110100%active
ITIXOXNOKVMBTE-UHFFFAOYSA-N110100%active
SGLIHNHGVBCTKU-UHFFFAOYSA-N110100%active
RYEPBHDKDSDCQV-UHFFFAOYSA-N101100%inactive
ORLXLKYURVKUJC-UHFFFAOYSA-N101100%inactive
ZJRLORBIIUEFCY-UHFFFAOYSA-N101100%inactive
LNLUHHXYUKPHKY-UHFFFAOYSA-N101100%inactive
WZYVNWKJPGKXRL-UHFFFAOYSA-N101100%inactive
FTMLRRDOVOHUFS-UHFFFAOYSA-N110100%active
RVXCQCJNPVTUQF-UHFFFAOYSA-N110100%active
HWAQFAYMDQZQES-UHFFFAOYSA-N110100%active
LSRMBMYSYMLMEU-UHFFFAOYSA-N110100%active
FUBOTVNFNSUKEY-UHFFFAOYSA-N101100%inactive
RFOUCZFAGRAPFU-UHFFFAOYSA-N110100%active
JGPQILYBQYCIDX-UHFFFAOYSA-N110100%active
BODDOMUCKPUVGY-UHFFFAOYSA-N101100%inactive
CNJKPUBUFXVNCF-UHFFFAOYSA-N101100%inactive
KCCHFUUIAZJPCS-UHFFFAOYSA-N202100%inactive
FQKVJCREIJRVNX-UHFFFAOYSA-N21150%exclude
YLWZWYDMYANSHU-UHFFFAOYSA-N21150%exclude
KPZFAFRIBLBLTA-UHFFFAOYSA-N101100%inactive
CFPKBGQZSYJRNG-UHFFFAOYSA-N21150%exclude
MHGBQBOLQZGDLP-UHFFFAOYSA-N101100%inactive
GIRDQOYFXWGMLW-UHFFFAOYSA-N202100%inactive
LMHXANVPOCTCND-UHFFFAOYSA-N21150%exclude
GFSUPLWNXMKMDH-UHFFFAOYSA-N21150%exclude
NGHIMGBPEPCNOT-UHFFFAOYSA-N21150%exclude
YFYHSMVMPADFTA-UHFFFAOYSA-N42250%exclude
GAEJFRRXRHOGOO-UHFFFAOYSA-N21150%exclude
XUYIOELVCRUWKB-UHFFFAOYSA-N21150%exclude
IMNPKIIYTUQSLC-UHFFFAOYSA-N101100%inactive
INHGUDXXUIVKLX-UHFFFAOYSA-N202100%inactive
CAJXAEQNBKVKTE-UHFFFAOYSA-N202100%inactive
NABMXRNHLTVSKG-UHFFFAOYSA-N21150%exclude
PNKZMKLBCXJMOP-UHFFFAOYSA-N63350%exclude
IVYRBVOBDZPTIK-UHFFFAOYSA-N21150%exclude
FCKYGPKVIITXMO-UHFFFAOYSA-N202100%inactive
UPTBAQYFWWXHPB-UHFFFAOYSA-N21150%exclude
NSSNPHNDZBWWAR-UHFFFAOYSA-N21150%exclude
VYOIHSHYYYZOMA-UHFFFAOYSA-N202100%inactive
NPPZPEXJTKIXER-UHFFFAOYSA-N21150%exclude
IYYJMJYGTSRZFT-UHFFFAOYSA-N21150%exclude
SQBWSWHAAIQVFL-UHFFFAOYSA-N21150%exclude
FNXVJFNFVIRKEU-UHFFFAOYSA-N101100%inactive
RDBFGHLYQLYGNT-UHFFFAOYSA-N21150%exclude
LZDRAGWKPJNEQC-UHFFFAOYSA-N21150%exclude
BADPLEONPHCMDZ-UHFFFAOYSA-N21150%exclude
MREFPWMRKNGHTG-UHFFFAOYSA-N202100%inactive
WXXWTZZAPUCLIM-UHFFFAOYSA-N202100%inactive
HHKGVQGXRGQBBA-UHFFFAOYSA-N101100%inactive
VRASPPLZZRUGFU-UHFFFAOYSA-N110100%active
IOQHKVXGXHYAJS-UHFFFAOYSA-N110100%active
YAZDYWJYFOMTQY-UHFFFAOYSA-N110100%active
GKLXUBYGZISONL-UHFFFAOYSA-N110100%active
VKRCGESNHINTGO-UHFFFAOYSA-N101100%inactive
OIRRXAJVSBXTIG-UHFFFAOYSA-N101100%inactive
QVNRUMIEALUOHI-UHFFFAOYSA-N101100%inactive
JMGKVLRBHUHFFV-UHFFFAOYSA-N101100%active
NVSGAXVEUPIOOQ-UHFFFAOYSA-N101100%inactive
OGZCHMBOZNMDQZ-UHFFFAOYSA-N110100%active
DAMJBUUVVWRAQN-UHFFFAOYSA-N101100%inactive
DVAYUYCZMIQXLC-UHFFFAOYSA-N101100%inactive
XHDJLFMWGGDHMB-UHFFFAOYSA-N101100%inactive
FMLPBXPSIJPCHY-UHFFFAOYSA-N101100%inactive
RKZNPODFSYTGAP-UHFFFAOYSA-N101100%inactive
IJAHGFUMVAVXQM-UHFFFAOYSA-N101100%inactive
CABJCPPEBOXLNC-UHFFFAOYSA-N101100%inactive
OGGVVKWMWABYPJ-UHFFFAOYSA-N101100%inactive
XMLWBUIPQKVCLK-UHFFFAOYSA-N101100%inactive
OVAXMETXFSJZJR-UHFFFAOYSA-N101100%inactive
OLLABBDDBLUFLY-UHFFFAOYSA-N101100%inactive
HNWOEIDVVRODCP-UHFFFAOYSA-N101100%inactive
KZNSDERJTMKOHV-UHFFFAOYSA-N101100%inactive
LIBMQZDDTQCBJD-UHFFFAOYSA-N101100%inactive
KFLRDJSBPGBGOL-JLRXKOEZSA-N101100%inactive
LNFBAYSBVQBKFR-UHFFFAOYSA-N101100%inactive
SZGHEGNWCACYLN-SJORKVTESA-N101100%inactive
PAOHWKCHWPLLOX-UXHICEINSA-N101100%inactive
OWOIXIRTYGMKDQ-MSOLQXFVSA-N101100%inactive
TYRRNKNTRGLDAB-UHFFFAOYSA-N101100%inactive
JZGAYLCRVBPMQG-MSOLQXFVSA-N101100%inactive
PKCIECLVWUJVCI-SJORKVTESA-N101100%inactive
TYRRNKNTRGLDAB-SJORKVTESA-N101100%inactive
WCIQHQDDKIZJND-MSOLQXFVSA-N101100%inactive
RNUSCQGPUILDPO-MSOLQXFVSA-N101100%inactive
BTWVWABAWDKQNJ-UHFFFAOYSA-N101100%inactive
SMOPKEHQPPXRSH-UHFFFAOYSA-N101100%inactive
OHNNRNYUHNGDNO-LSDHHAIUSA-N101100%inactive
WAAWETUDFSIYSD-UHFFFAOYSA-N101100%inactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N101100%inactive
NWXGFDVFXJMUDD-UHFFFAOYSA-N101100%inactive
TXEBNKKOLVBTFK-UHFFFAOYSA-N101100%inactive
FPLYXYDSEPGNHS-UONOGXRCSA-N101100%inactive
FSAPXEJFAWOTKO-UHFFFAOYSA-N101100%inactive
NDNLATIKQBVEQQ-UHFFFAOYSA-N101100%inactive
MHBAZXJUDZFMFF-UHFFFAOYSA-N101100%inactive
SLFFKTMXFBIVIA-UHFFFAOYSA-N101100%inactive
QMEDNEYWSPIHTH-UHFFFAOYSA-N101100%inactive
YSXMSGJFZINEEZ-UHFFFAOYSA-N101100%inactive
VPFOKEYECQYGJV-UHFFFAOYSA-N101100%inactive
DXCIBUPROMUQLA-UHFFFAOYSA-N101100%inactive
UFWDODPQTYHRKT-UHFFFAOYSA-N101100%inactive
JTGRBZUCDOIAAL-UHFFFAOYSA-N101100%inactive
ZMNWFTYYYCSSTF-SOAUALDESA-N101100%inactive
IGDFNCLISYKTLQ-UHFFFAOYSA-N101100%inactive
IOZRQIXIPZEKNW-UHFFFAOYSA-N101100%inactive
CUPLTRAPYIXFAX-UHFFFAOYSA-N101100%inactive
DVRSTRMZTAPMKO-UHFFFAOYSA-N101100%inactive
DGUSFVFTIHATAT-UHFFFAOYSA-N101100%inactive
JLIDQWKTZPUAMJ-UHFFFAOYSA-N101100%inactive
JOEQBUIAUWMVDT-UHFFFAOYSA-N101100%inactive
QTWZRRQQWNQCMR-UHFFFAOYSA-N101100%inactive
WJFHDSLGZITKRZ-UHFFFAOYSA-N101100%inactive
HBCPKSWKTFFBIK-UHFFFAOYSA-N101100%inactive
GMVQPWCWWLPOQT-FQEVSTJZSA-N101100%inactive