P53350 PLK1


Group: Other
Family: PLK
PDB Structure Num: 12
FDA approved drugs from DrugBank: Fostamatinib






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
QDLHCMPXEPAAMD-QAIWCSMKSA-N101100%inactive
MNMQBQOLMHVBJT-UHFFFAOYSA-N101100%inactive
HEUHMWCGNUTYFR-SOVKOMHZSA-N101100%inactive
AFSDNFLWKVMVRB-UHFFFAOYSA-N101100%inactive
SXNJFOWDRLKDSF-STROYTFGSA-N330100%active
XQVVPGYIWAGRNI-JOCHJYFZSA-N660100%active
VQIOLOBSXRKEAP-KIUCONSDSA-N101100%inactive
LNHXIPPBAPMRIE-AYTHIJHQSA-N110100%active
UQVVKCSRCFXOOS-KIUCONSDSA-N110100%active
WGXULIDEUYMONG-KIUCONSDSA-N101100%inactive
OYUCIHXKLQGOKP-WYEJJTDISA-N101100%inactive
CZPWZRXIYDNNLI-BKXCAEITSA-N110100%active
ZDQJNYLFGPXANH-BKXCAEITSA-N550100%active
UIYQCJDQBRUFEV-FALOATQWSA-N303100%inactive
FXFITXFZTUYDTA-UHFFFAOYSA-N303100%inactive
IYLBMSHZRRWSRM-FALOATQWSA-N202100%inactive
VRWFLNVDDMVVDA-OFMCOEKFSA-N101100%inactive
XEGSWNKCRGYRFG-HEPSPIFKSA-N101100%inactive
QPBYPJKNTKPWHP-XRSOISPESA-N110100%active
QECCEBUDDKKVOA-KQFQEUIISA-N101100%inactive
DDUIKWXPFWIAGL-OMAZYLPNSA-N101100%inactive
OORPAHIABJKOQZ-QMBSKNLRSA-N101100%inactive
DEHXVDBTGRNEJG-GSESMZNDSA-N101100%inactive
JLXBABLXNALFOP-IHNFJAPISA-N101100%inactive
RBXLZSWSJTUVKC-LJAQVGFWSA-N110100%active
IVRPFXYSCCXTAK-MUUNZHRXSA-N110100%active
GWRSATNRNFYMDI-UHFFFAOYSA-N110100%active
WYSOLHCQRQBXQP-UHFFFAOYSA-N110100%active
RXDSAQWDJRAMCT-UHFFFAOYSA-N110100%active
BAVKHKJJAGWXBX-UHFFFAOYSA-N110100%active
AEWBIFRPDTZPLO-UHFFFAOYSA-N110100%active
JMBATVPHKFZTAF-UHFFFAOYSA-N110100%active
WQQPBXGJFFKXKX-UHFFFAOYSA-N110100%active
JFRNFMQDZRWAQB-UHFFFAOYSA-N110100%active
DJNZZLZKAXGMMC-UHFFFAOYSA-N110100%active
QEIJYXMTALGXJH-GDLZYMKVSA-N110100%active
QEIJYXMTALGXJH-LJAQVGFWSA-N110100%active
DWBXNQKRJAOIHK-NRFANRHFSA-N110100%active
DWBXNQKRJAOIHK-OAQYLSRUSA-N110100%active
RBXLZSWSJTUVKC-GDLZYMKVSA-N110100%active
WFYIXLNYITUPPQ-QGZVFWFLSA-N101100%inactive
LBJBUWVRDHIUEP-UHFFFAOYSA-N101100%inactive
YUWWKWVVBFASIG-UHFFFAOYSA-N101100%inactive
RJCQITTXWSWFFO-UHFFFAOYSA-N101100%inactive
ZQQFEJKKQWPBQA-UHFFFAOYSA-N101100%inactive
JMDRAMDTWLAOHD-GOSISDBHSA-N110100%active
PMMISILPBLQWSZ-GFCCVEGCSA-N101100%inactive
GNFVJCMQLYMYRH-MRXNPFEDSA-N101100%inactive
KOKNYBBQIVDZCK-OAHLLOKOSA-N110100%active
XDUIHJCDFMNCIS-OAHLLOKOSA-N101100%inactive
RHIJMDNVEPLDED-UHFFFAOYSA-N110100%active
WKIWJYRJQNQEGF-MRXNPFEDSA-N101100%inactive
UMJFDLYATACWKW-DLBZAZTESA-N110100%active
UMJFDLYATACWKW-IAGOWNOFSA-N110100%active
HXPKCEXQOBXOIS-DLBZAZTESA-N101100%inactive
ZJJBLPXVAOPPAR-UHFFFAOYSA-N101100%inactive
QWAKOUIKNVQHES-UHFFFAOYSA-N101100%inactive
SQHOHRAPERDRPS-UHFFFAOYSA-N101100%inactive
HKSMOPLPIGGMTK-QGZVFWFLSA-N101100%inactive
DDHRKINLNCDPNG-MRXNPFEDSA-N101100%inactive
QCJIMVKECGDPPA-UHFFFAOYSA-N101100%inactive
RVEBOFKFYDCQPT-QGZVFWFLSA-N101100%inactive
JMVCDNFYMJCUDW-MRXNPFEDSA-N101100%inactive
RJBBMLHRKBGRBY-MRXNPFEDSA-N101100%inactive
NILXCNICWMPUMM-CQSZACIVSA-N110100%active
PBCXNVUBDXBJNG-WCQYABFASA-N101100%inactive
CPDRDZZZFNTJCE-GFCCVEGCSA-N101100%inactive
XNXPWGGHJWESTI-UHFFFAOYSA-N101100%inactive
ABRWDZBHBOWGSY-WCIBSUBMSA-N101100%inactive
VHVCSZNJCUZDOG-LCYFTJDESA-N101100%inactive
QJJAFCLEWYTXRC-XFXZXTDPSA-N101100%inactive
PXBQEMZXNXEANC-YRNVUSSQSA-N101100%inactive
HKGXDXUDOHQKPM-JYRVWZFOSA-N101100%inactive
MPFUDUPAOWHBRQ-NTUHNPAUSA-N101100%inactive
HOOFEYTZWSBHNO-WLRTZDKTSA-N101100%inactive
HOOFEYTZWSBHNO-ACAGNQJTSA-N101100%inactive
LFKWPZDAYPDIKU-WLRTZDKTSA-N101100%inactive
KFZCNVWXULQFPN-MKMNVTDBSA-N101100%inactive
MDYWOSMFBZFSBX-MKMNVTDBSA-N101100%inactive
PLAOAGFXNCEZMZ-LCYFTJDESA-N101100%inactive
LMXYVLFTZRPNRV-KMKOMSMNSA-N101100%inactive
AHNFXMBOWJVAPB-FUHWJXTLSA-N101100%inactive
IREYRQPUBOQACQ-UHFFFAOYSA-N101100%inactive
HTCVSLIHSFBUEL-UHFFFAOYSA-N101100%inactive
REFJWTPEDVJJIY-UHFFFAOYSA-N101100%inactive
ACOQUBGHQYPJFN-NZZVAQPWSA-N101100%inactive
VXQUGYOYJDITTO-KNSMUJDWSA-N101100%inactive
UGEGMLHKJYPRKJ-JLHYYAGUSA-N101100%inactive
YGPQMFXMKKHCNZ-SOFGYWHQSA-N110100%active
UWCNNPLPNWIHHP-VMPITWQZSA-N110100%active
DGVGLURAKIWTCE-QPJJXVBHSA-N101100%inactive
AAMGHFYBPZUVNQ-FPYGCLRLSA-N101100%inactive
XTYDCDUVSAESPJ-FPYGCLRLSA-N101100%inactive
FAXITRGBEHCSIB-RMKNXTFCSA-N101100%inactive
HRESQKRNIZIAQQ-RUDMXATFSA-N110100%active
MJJUKTUICBQNBI-FPYGCLRLSA-N110100%active
KOGRIKJYGMBXFL-RMKNXTFCSA-N110100%active
KRHMAJOTJVOLBI-VXLYETTFSA-N101100%inactive
HCBULGQMULJTCM-RIYZIHGNSA-N101100%inactive
WQKKJLNOWMZBOW-UHFFFAOYSA-N110100%active
OWBFCJROIKNMGD-BQYQJAHWSA-N110100%active
KEQHJBNSCLWCAE-UHFFFAOYSA-N101100%inactive
MHSBQWAPDZNAST-UHFFFAOYSA-N101100%inactive
JZGUHPFQSABXEO-UHFFFAOYSA-N101100%inactive
FJZAHNJWHBXOJX-UHFFFAOYSA-N101100%inactive
ZIVMVDLFRZESTI-UHFFFAOYSA-N101100%inactive
FZBGHMKUJJAGBT-UHFFFAOYSA-N101100%inactive
XATBCOLGACXQQM-UHFFFAOYSA-N101100%inactive
HNOLYVYDGDGIDD-UHFFFAOYSA-N110100%active
VFXXPAORMIDACS-UHFFFAOYSA-N110100%active
IUESHCGRXYXZSP-UHFFFAOYSA-N101100%inactive
JHYRCHZGDMGSLM-UHFFFAOYSA-N101100%inactive
OIKYUBXQDWHHJC-UHFFFAOYSA-N101100%inactive
OQQFXVWSINWEED-UHFFFAOYSA-N101100%inactive
UKDYPCZCLRCOMP-HXUWFJFHSA-N110100%active
SWTRIZHCIUWGAU-UHFFFAOYSA-N110100%active
OXPLZKSKLWBEIM-UHFFFAOYSA-N110100%active
TUWAYASUNDRSML-UHFFFAOYSA-N110100%active
VEFDUZNTHFBSFU-UHFFFAOYSA-N110100%active
QHLVBNKYJGBCQJ-UHFFFAOYSA-N110100%active
DFKJNGVBNCASDM-UHFFFAOYSA-N110100%active
VPWDLLHGBJTELF-UHFFFAOYSA-N110100%active
OCPMRHZHACWECI-UHFFFAOYSA-N110100%active
IWNBRVJHAXKTLL-UHFFFAOYSA-N110100%active
QROBXWMBDYEVNI-UHFFFAOYSA-N110100%active
RBYMMVRBIIJFHH-UHFFFAOYSA-N110100%active
ZPROSCYPYBVWCA-UHFFFAOYSA-N110100%active
NIYZKZFROMUIEF-UHFFFAOYSA-N110100%active
ZMMZXGLECYSZEP-UHFFFAOYSA-N110100%active
HWLKVHNUFPRSIJ-UHFFFAOYSA-N110100%active
FJECSOOLAWUZAB-UHFFFAOYSA-N101100%inactive
YISMQBFJYDFMAL-MCGZHFTPSA-N101100%inactive
UEMYVTYHECWXSR-WDZFZDKYSA-N101100%inactive
GQULUVWAOIVUQB-UHFFFAOYSA-N110100%active
FSCIFRALUGPNIF-VUIPXDDYSA-N110100%active
SSGQBUPRSFPFIB-GHOWNLRVSA-N110100%active
ACUJSWPHFSMCON-KITDGBJQSA-N21150%exclude
KJQNIUMZTBTNPM-TYYMDPTCSA-N202100%inactive
UPWFDMAFUHNQNM-XIKJUOIESA-N110100%active
NDZJFAYZPBTTDL-IQJHCYRHSA-N202100%inactive
KSYUJQDWOGQQIP-NXWKYJJNSA-N110100%active
QINOMHBLNDVOTP-GXQKTUKWSA-N21150%exclude
WXWYPJSPBYNUSZ-IRBCDZGCSA-N110100%active
RZLIRASVOYQCEI-VPGGRGEMSA-N110100%active
YDADPNOVOQSBSB-LPQCQSQESA-N110100%active
LYLANQFTXJWIGY-SWLZGSTDSA-N110100%active
VWTMBJNORZHGHE-ICMBXEKGSA-N110100%active
XDRHCUWKZRZSEP-CQKJNDIKSA-N330100%active
VBUBVQOQXYMYMF-KJHGNAGRSA-N110100%active
ZPKPKCOLWJOVJV-ZTHSRUGTSA-N110100%active
GXROUISBNDMFKO-WTZADEQLSA-N110100%active
NDKOLPRDQQUJPD-UHFFFAOYSA-N202100%inactive
CMOJHDQJJPIVEC-MNDPQUGUSA-N101100%inactive
XLFNLJYGUOLEJS-SFHVURJKSA-N101100%inactive
AWYSFWYRQPHWJL-JOCHJYFZSA-N110100%active
XFQQKFNFMHVKGP-XMMPIXPASA-N110100%active
NVZUHQUNIGVGBQ-HSZRJFAPSA-N110100%active
KRKASDMDACZHLR-XMMPIXPASA-N110100%active
UJEXFMKGBVBXPF-XMMPIXPASA-N110100%active
XKVZTXMZBWFWRQ-RUZDIDTESA-N110100%active
IYWCICTYSWDBDQ-XMMPIXPASA-N110100%active
GHMBRNIPQXNYFY-JOCHJYFZSA-N110100%active
LZDAATYWWSHULX-HXUWFJFHSA-N110100%active
RBFXWJWEHFNLDF-HSZRJFAPSA-N110100%active
CBNBACZYZVMFBW-JOCHJYFZSA-N110100%active
CKAZLPSHMQDEHE-OYPUMOIUSA-N110100%active
TYJHZOFBUGXDFG-XMMPIXPASA-N110100%active
UMYZHTXQBNEZNF-JOCHJYFZSA-N110100%active
WQQABBZFVHSXMU-FWZUBCPGSA-N220100%active
SHZJITZSGHNGAS-USJNNXEMSA-N220100%active
STDVQZAYBMZKHW-SMKGIDQESA-N21150%exclude
KSMYGTHXVJXRTI-UONILZFISA-N220100%active
COQMBZDAQWGIGH-UHFFFAOYSA-N101100%inactive
MLSDGZDBIVDXEE-UHFFFAOYSA-N101100%inactive
WIVJBVXMFDYZEO-UHFFFAOYSA-N101100%inactive
LKKGYKDFEPORRK-UHFFFAOYSA-N101100%inactive
UPGDJDYZVVFRFD-UHFFFAOYSA-N101100%inactive
KASGWSVWRRHWBU-UHFFFAOYSA-N101100%inactive
QHPKKGUGRGRSGA-UHFFFAOYSA-N101100%inactive
PZPCKANQRXHUSX-UHFFFAOYSA-N101100%inactive
YYZTVTZCYVZGRB-UHFFFAOYSA-N110100%active
RNXPIGAWEIQILT-UHFFFAOYSA-N110100%active
JALCTFDLDSFBBC-UHFFFAOYSA-N101100%inactive
XKFTZKGMDDZMJI-HSZRJFAPSA-N101100%inactive
SWIVJTVGOIXUKC-MRXNPFEDSA-N110100%active
MOSNATYSIYEVTF-MRXNPFEDSA-N110100%active
VVQWZQWJWMTPJY-QZTJIDSGSA-N110100%active
SLGRRBVHGIPHNQ-OAHLLOKOSA-N110100%active
HLHNFPFYQRRGPP-MSOLQXFVSA-N110100%active
HLHNFPFYQRRGPP-QZTJIDSGSA-N110100%active
RUTCIZOQGCWURK-UHFFFAOYSA-N101100%inactive
RLARTPHANIERPF-AWEZNQCLSA-N101100%inactive
NTAIRXFACXVUQO-AWEZNQCLSA-N110100%active
RMKFZACOOVWLAE-HNNXBMFYSA-N101100%inactive
CYRHCHWHTHQZAV-INIZCTEOSA-N110100%active
MMGKIHLBFPJYJL-HNNXBMFYSA-N110100%active
HMLWZSKONNDQRL-LBPRGKRZSA-N101100%inactive
KVJXBCZPOFTDAU-AWEZNQCLSA-N110100%active
RRBCORZOVOSGLG-CKDBGZEDSA-N101100%inactive
IDWMLMNMILZSML-AWEZNQCLSA-N101100%inactive
OKIPMNUDSPZOMT-HNNXBMFYSA-N101100%inactive
ZOIMQOAMAULHEL-MYJWUSKBSA-N101100%inactive
DAAGOCSHXCDWDY-ZDUSSCGKSA-N110100%active
CQYPOADQLJEUBB-ZDUSSCGKSA-N101100%inactive
QNYZHMLWZSRWRH-ZDUSSCGKSA-N101100%inactive
DJNPBANWRKSHQM-HNNXBMFYSA-N101100%inactive
XZPCSXAQYZGHKR-QPLCGJKRSA-N101100%inactive
XZXHXSATPCNXJR-ZIADKAODSA-N101100%inactive
DUZZUNRKDFGPSJ-IZHYLOQSSA-N101100%inactive
ORKOHXAJFGRZCL-LCYFTJDESA-N101100%inactive
ZXFBTQCKAZQQFA-CNIJLMKKSA-N101100%inactive
USFQLAVWHQCNDG-AYEIPMSGSA-N101100%inactive
OZROZYIBIZOAQQ-DLBXBJKMSA-N101100%inactive
XXLLTYLTCDARFZ-OHSNSYSLSA-N101100%inactive
GKFHBWBDOADOEV-HFOUWSASSA-N101100%inactive
RAIDHOLJIAWOMY-DKQGWWAXSA-N101100%inactive
MDPPOIXSNMVHOD-FBPKMIEBSA-N101100%inactive
DGOKKNPUISUUGY-UHFFFAOYSA-N101100%inactive
LKXFSTAQMOENSC-UHFFFAOYSA-N101100%inactive
QPOURHROVVCOHC-UHFFFAOYSA-N101100%inactive
LNFBAYSBVQBKFR-UHFFFAOYSA-N101100%inactive
NZCHGHMPHKCWLR-UHFFFAOYSA-N101100%inactive
QHUDPFOODLMGQO-UHFFFAOYSA-N101100%inactive
PUJKNBHSGMNWBW-UHFFFAOYSA-N101100%inactive
RIOJOTOJNAHBST-UHFFFAOYSA-N101100%inactive
RCTLMZOWMCIZPV-UHFFFAOYSA-N101100%inactive
UFRMEDNDGZCHLF-MRXNPFEDSA-N101100%inactive
AxitinibRITAVMQDGBJQJZ-FMIVXFBMSA-N101100%inactive
FOMWYZMFUGYYLZ-ADFPNGHDSA-N101100%inactive
BPGUPPRJBLLMOX-JDCCHMEXSA-N101100%inactive
CPIOXRCBBSICIO-SLUIUKIVSA-N101100%inactive
OLRQMHGOBAYXHZ-FPQBULDBSA-N101100%inactive
ZGEQGZFSJZJWAR-JNJFRLMHSA-N101100%inactive
CZFUYZPXZGGWKC-SRQUHQSVSA-N202100%inactive
VFYXAFQACZHFRL-NHSDSWEZSA-N101100%inactive
QDBKDMHYYVPUJY-UJPRRALESA-N101100%inactive
DOLNBRDFBGDLQN-VGKQJACHSA-N101100%inactive
YKIVNICLNFURQO-NHSDSWEZSA-N101100%inactive
YJKHNFBXHIHRMJ-WRMRRPGHSA-N101100%inactive
HCLJFCCORISDCX-NLUXTTPZSA-N101100%inactive
UPAQROHCJDLJNE-JBFZHCRBSA-N101100%inactive
FQWPBCFJZAKNEQ-CBVNATGFSA-N101100%inactive
GBUDRABUNBYJKG-WWAWLHJKSA-N101100%inactive
GKBCILCXUSENIW-XGICHPGQSA-N101100%inactive
DMFNFAMMDAVMRL-XGICHPGQSA-N101100%inactive
JLCLRTONUBKGKP-WZUFQYTHSA-N101100%inactive
ULXYLHILBRICFA-WLRTZDKTSA-N101100%inactive
UXFLFGRXPDAOOG-GIDUJCDVSA-N101100%inactive
QFMBWTHKAIYHLD-GIDUJCDVSA-N101100%inactive
PZBSSTRXBNWBNX-UHFFFAOYSA-N101100%inactive
WTFXMLVITCJWNE-UHFFFAOYSA-N101100%inactive
KYBALIQJYSWGLI-UHFFFAOYSA-N101100%inactive
ATQVAIUSAHRLDF-KSVBPBMVSA-N101100%inactive
RGIXMSXCHQWNPC-UHFFFAOYSA-N101100%inactive
SEVGOOROBLVJGK-UHFFFAOYSA-N101100%inactive
XGSCWZVQRNHENL-RMKNXTFCSA-N101100%inactive
UKZRGBUTBINTPD-LOSJGSFVSA-N101100%inactive
PNMQDIXULZYDDT-UHFFFAOYSA-N101100%inactive
BUMGKNPRCXMAGM-FVOFJUMPSA-N101100%inactive
NZBZBQUHFXSFOR-VXPCJWDYSA-N101100%inactive
JAHXQCZCZURPTI-UHFFFAOYSA-N101100%inactive
JBZRAEUHDPMQSF-UHFFFAOYSA-N101100%inactive
CGXHFSJDSWAEMT-UHFFFAOYSA-N101100%inactive
OWLAKERMHYDWTB-UHFFFAOYSA-N101100%inactive
FGNQVZZMORDWIZ-UHFFFAOYSA-N101100%inactive
GIAVVFIPFBOBRR-UHFFFAOYSA-N101100%inactive
QPVNTDBWWRFMIC-UHFFFAOYSA-N101100%inactive
QUYGYUVUHYMMRW-UHFFFAOYSA-N101100%inactive
DADASRPKWOGKCU-FVTQAUBDSA-N101100%inactive
ARYVAQSYRLZVQD-UHFFFAOYSA-N101100%inactive
VBYMFAOTZHNONG-UHFFFAOYSA-N101100%inactive
WAAWETUDFSIYSD-UHFFFAOYSA-N101100%inactive
VRQXRVAKPDCRCI-ZNMIVQPWSA-N101100%inactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N202100%inactive
AECDBHGVIIRMOI-GRGXKFILSA-N101100%inactive
YXLQJZQRBVGUCM-ZVDOUQERSA-N101100%inactive
WNYKGJHEQVIFGL-OAHLLOKOSA-N101100%inactive
XTJZKALDRPVFSN-HNNXBMFYSA-N101100%inactive
OSAWFUCUZJNEID-CQSZACIVSA-N101100%inactive
MELHJKUYOBXOER-UHFFFAOYSA-N101100%inactive
OJLPXQRQXJPIKO-UHFFFAOYSA-N101100%inactive
DCRJMZNHTPDFNQ-UHFFFAOYSA-N101100%inactive
QEWMJARXNKOXMM-UHFFFAOYSA-N101100%inactive
ZCJZGTHJIXYVGG-UHFFFAOYSA-N101100%inactive
ALIXTVBPMHJTAF-UHFFFAOYSA-N101100%inactive
CAVFEAKOYPWCSA-UHFFFAOYSA-N101100%inactive
SGCQJCPNXKHNPH-UHFFFAOYSA-N101100%inactive
GSCAIAFNYPEEIT-UHFFFAOYSA-N101100%inactive
KMIHVDIUSIWJBR-UHFFFAOYSA-N101100%inactive
MWEIZALZQKSIDX-UHFFFAOYSA-N101100%inactive
ORWCFWCLFTZXTR-UHFFFAOYSA-N101100%inactive
UJXSEZDSHGPMOE-UHFFFAOYSA-N101100%inactive
MNXLTLCOWQQAKN-UHFFFAOYSA-N101100%inactive
CFCOQYROFLFNOU-UHFFFAOYSA-N101100%inactive
UWHWQUTVFLDMPJ-UHFFFAOYSA-N101100%inactive
CZGMEOAMQWAJOY-UHFFFAOYSA-N101100%inactive
BOJMKEOOGVQEAQ-HNNXBMFYSA-N101100%inactive