P51812 RSK2


Group: AGC
Family: RSK
PDB Structure Num: 5
FDA approved drugs from DrugBank: Fostamatinib






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
RHBGODQVOKDULK-UHFFFAOYSA-N101100%inactive
RDGQRZYRTFWBJR-UHFFFAOYSA-N101100%inactive
UJAUSTYSRUCHNY-UHFFFAOYSA-N220100%active
SPOWSXDVDODVEW-UHFFFAOYSA-N220100%active
JBOKTWNEIMBJNQ-UHFFFAOYSA-N220100%active
UERCXNOQFSTSOY-UHFFFAOYSA-N220100%active
JMEYCQCGWJJILQ-UHFFFAOYSA-N220100%active
PXRIUZVVLPVSSH-UHFFFAOYSA-N21150%exclude
YVUHNKZPGGBYDH-UHFFFAOYSA-N220100%active
RXYDOJKKUXRPAA-UHFFFAOYSA-N220100%active
WKUUMSASAHOWGZ-UHFFFAOYSA-N220100%active
WIICYVHPNFINMO-UHFFFAOYSA-N220100%active
NRGYMIVHSWOTKI-UHFFFAOYSA-N220100%active
HZZNLCVNOOMGDD-UHFFFAOYSA-N220100%active
YARFNYLGLQVPEB-UHFFFAOYSA-N21150%exclude
KAKNBLVUBRXYQD-UHFFFAOYSA-N220100%active
GVDISXKMIUKGIP-UHFFFAOYSA-N220100%active
QYLAYPRSSJNQDC-UHFFFAOYSA-N220100%active
VCZQSUBZCZZLAX-UHFFFAOYSA-N220100%active
WMGGYIKBPUVPFM-UHFFFAOYSA-N220100%active
ZHMXXVNQAFCXKK-QGZVFWFLSA-N220100%active
ZHMXXVNQAFCXKK-KRWDZBQOSA-N220100%active
LQZKYXLZCLMOGP-UHFFFAOYSA-N220100%active
LAJAFFLJAJMYLK-CVOKMOJFSA-N110100%active
SVXJIKFFHBDTNV-SFQUDFHCSA-N110100%active
IKLGYJACVCXYIL-UHFFFAOYSA-N220100%active
PRMVLMCLSDUYOK-ODHHTFEASA-N110100%active
YKEOPYUONVHGAZ-JPJNWVEQSA-N101100%inactive
KJCRKINUZWFECN-QXKHQJIESA-N101100%inactive
XDTPAAMXVSEUMQ-IMLMFSNGSA-N110100%active
LYPFUSXIPAESSO-JRQRPHQWSA-N101100%inactive
KJNVQQRKZXSWGI-WGXSRGGHSA-N101100%inactive
HDCQFGSWWKAJHS-UDKWMEDXSA-N101100%inactive
SXOZSDJHGMAEGZ-IGKKHSBFSA-N43175%exclude
XLYVQVWMTOLDNL-ZROIWOOFSA-N21150%active
RINGOEHWKXCHGN-GDNBJRDFSA-N101100%inactive
DINXQJVLLOMREI-NVNXTCNLSA-N101100%inactive
YKPCAIZGCTXESO-CLFYSBASSA-N101100%inactive
WSOJBINOLIOJTD-NTMALXAHSA-N101100%inactive
PGZGBDVILWVGSF-FLIBITNWSA-N202100%inactive
LQIWKQNFITUIPZ-YRNVUSSQSA-N101100%inactive
CBYUHHGMVIHGFQ-YRNVUSSQSA-N101100%inactive
VSEGODXJTWWVIT-YRNVUSSQSA-N101100%inactive
KLJVDMAOKMSBQX-UHFFFAOYSA-N101100%inactive
YPNCCYRKEHPJMN-LJQANCHMSA-N101100%inactive
LLFRXYFZGCTTDG-OTGJNIAMSA-N110100%active
HEDQIXPQCXBXDD-HZQSEOSJSA-N101100%inactive
WADXCMSONJVPKX-LTBIHHBXSA-N101100%inactive
OTPCQHIGGWABCT-CVOKININSA-N101100%inactive
FHGTUVGVZRNUDB-UHFFFAOYSA-N110100%active
RYNUCFRWRKDYTQ-UHFFFAOYSA-N110100%active
NKCQURNGRKMMNF-UHFFFAOYSA-N101100%inactive
HSHRVAFOSVHQNQ-UHFFFAOYSA-N110100%active
LKJIWFIGQMHDPR-UHFFFAOYSA-N110100%active
FTUOTWYRSQTGOK-UHFFFAOYSA-N110100%active
VTDTXABIZXUXME-UHFFFAOYSA-N110100%active
WQBTWNKSFDRALJ-UHFFFAOYSA-N110100%active
VACMZWAHKWHHMN-UHFFFAOYSA-N110100%active
OGRWLDHVLHSNOM-UHFFFAOYSA-N101100%inactive
HRIBPTNPPPEBMO-UHFFFAOYSA-N101100%inactive
RXJKIHBSKCIXKE-UHFFFAOYSA-N110100%active
CZIQZFRYLZOTAU-UHFFFAOYSA-N110100%active
SRNVWQXDZWXKFC-UHFFFAOYSA-N110100%active
SKGOKFXHVKRTIW-UHFFFAOYSA-N110100%active
JXGRDWXLVXGFGC-UHFFFAOYSA-N110100%active
AJGHEMDMZKKTSJ-UHFFFAOYSA-N110100%active
WEXZHJRBQNKEKT-UHFFFAOYSA-N110100%active
UUTIVRONEJLBDK-UHFFFAOYSA-N110100%active
LNVRALGTJWRQTK-UHFFFAOYSA-N110100%active
RTECQFROUMPSQG-UHFFFAOYSA-N110100%active
VAMWJMVATUYTLB-UHFFFAOYSA-N110100%active
IKUFKDGKRLMXEX-UHFFFAOYSA-N110100%active
YUYJEQHNWKQNBT-UHFFFAOYSA-N110100%active
NKBWZEGVHYSODY-UHFFFAOYSA-N110100%active
FWJNKYPUQRBACL-UHFFFAOYSA-N101100%inactive
ZPBALWYVPVVNDT-UHFFFAOYSA-N110100%active
GIFPFLKKKQLPLV-UHFFFAOYSA-N110100%active
RTHBKFCPLFHNBB-UHFFFAOYSA-N110100%active
PBZUKXQEJRTGRV-UHFFFAOYSA-N110100%active
HPQKQSNTXXYIDR-UHFFFAOYSA-N110100%active
SZXVKXAUZJIMFQ-UHFFFAOYSA-N110100%active
OEOITLSQKKJYKY-UHFFFAOYSA-N110100%active
KDSPNDQAEMFZQR-UHFFFAOYSA-N110100%active
DTEKTGDVSARYDS-LLVKDONJSA-N110100%active
TWUMJNHHODMHNL-UHFFFAOYSA-N110100%active
ZAAULFKSCDOLLO-UHFFFAOYSA-N110100%active
NTXOERDSELUUJC-UHFFFAOYSA-N101100%inactive
XUAKNRZAHPCZNV-UHFFFAOYSA-N110100%active
HIWDEEKFVOBEDG-UHFFFAOYSA-N110100%active
SMUQHDGUBPGZGE-UHFFFAOYSA-N101100%inactive
NOLQEYVCYRCPPK-UHFFFAOYSA-N110100%active
GEAJTWHHUPQLRH-UHFFFAOYSA-N101100%inactive
VIXLRYPHJBBDMB-UHFFFAOYSA-N101100%inactive
VFOVHOQMPWWNPV-UHFFFAOYSA-N110100%active
UNRWZBUXURMJLA-UHFFFAOYSA-N110100%active
DBQAJQQGPQIDLD-UHFFFAOYSA-N101100%inactive
IUBOVMXHGBTLME-UHFFFAOYSA-N101100%inactive
BNGKFHKLNDIATR-UHFFFAOYSA-N110100%active
KIVVSMMKIIIXEN-UHFFFAOYSA-N101100%inactive
HGWRPHQJLMJBQA-UHFFFAOYSA-N110100%active
HXTSCEKORFMGBI-UHFFFAOYSA-N110100%active
IBUYZUJUVMHXAU-UHFFFAOYSA-N110100%active
XPXROBNEPUYDHT-UHFFFAOYSA-N110100%active
SMGYOERWRLLOJT-UHFFFAOYSA-N110100%active
ANDKZPJYPPFDOM-UHFFFAOYSA-N101100%inactive
MIBQXOPDHBSXEI-UHFFFAOYSA-N101100%inactive
SUWROSUZAZIMBS-UHFFFAOYSA-N101100%inactive
CTPVTASKZQBESS-UHFFFAOYSA-N110100%active
JSGGVCXEKFWRSW-UHFFFAOYSA-N110100%active
JGGFTDCGSPWVHI-UHFFFAOYSA-N110100%active
GXOLWQVEFZJSDG-UHFFFAOYSA-N110100%active
ZBPWYWRJCWAYEQ-UHFFFAOYSA-N110100%active
HFKVSRQGYCGTCO-UHFFFAOYSA-N110100%active
YBDVSJKTAWTRHQ-UHFFFAOYSA-N110100%active
KSLDAMNDQVGQHI-UHFFFAOYSA-N110100%active
BVXJEHLFTPAGNE-UHFFFAOYSA-N110100%active
HHBAYTAFBOSZPX-UHFFFAOYSA-N110100%active
ZDLIZWHPESZXOR-UHFFFAOYSA-N110100%active
ZISHPQSNRHWEJX-UHFFFAOYSA-N110100%active
GXLSDFNOALILGU-UHFFFAOYSA-N110100%active
DPQHQAXUONFMQP-UHFFFAOYSA-N110100%active
OBKXLPJQBTZBMA-UHFFFAOYSA-N110100%active
JKXDDXLLFULDSB-UHFFFAOYSA-N110100%active
QEQUMZRCCUEIIJ-UHFFFAOYSA-N110100%active
IEWJUSIVLMUWOD-UHFFFAOYSA-N110100%active
VGBPXKNBWHOARX-UHFFFAOYSA-N110100%active
HIYHAWWDKKWHQY-UHFFFAOYSA-N110100%active
IIDUHZAGWFEQBW-UHFFFAOYSA-N110100%active
BLIQORTUYKIMFR-UHFFFAOYSA-N110100%active
OJPHUPWPAOYDSF-UHFFFAOYSA-N110100%active
VHYKGAUCYCNUBF-UHFFFAOYSA-N110100%active
FVUHABBLIJXZMN-UHFFFAOYSA-N110100%active
MISDLVFAYWWZLG-UHFFFAOYSA-N110100%active
XDFUUIPECUWQQZ-UHFFFAOYSA-N110100%active
PNSOZKZGPSQHSN-UHFFFAOYSA-N110100%active
UFFQKOHHXSMIRW-UHFFFAOYSA-N110100%active
RPBYOOGHPJSODY-UHFFFAOYSA-N101100%inactive
YHWMUAMXBJBKPC-UHFFFAOYSA-N101100%inactive
NQXBMUAFKYZLNH-UHFFFAOYSA-N101100%inactive
HNSNQBPXQBNWAY-UHFFFAOYSA-N110100%active
IFLNKMNSCZBCLT-UHFFFAOYSA-N110100%active
IIHMKUHCZGYMCV-UHFFFAOYSA-N110100%active
BYNBSGRVCINSBK-UHFFFAOYSA-N101100%inactive
GRKDQSJJVVIXFN-CQSZACIVSA-N110100%active
GRKDQSJJVVIXFN-AWEZNQCLSA-N110100%active
UHXBEOZTLFAXRQ-CABCVRRESA-N110100%active
UHXBEOZTLFAXRQ-GJZGRUSLSA-N110100%active
MOAVQHGMQJPAOO-LBPRGKRZSA-N110100%active
GNBSFKOHIIYQLM-GFCCVEGCSA-N110100%active
GNBSFKOHIIYQLM-LBPRGKRZSA-N110100%active
MOAVQHGMQJPAOO-GFCCVEGCSA-N110100%active
ULXCPSCTMQCILD-UHFFFAOYSA-N110100%active
BYNSQSZIQPYTMV-UHFFFAOYSA-N110100%active
JSMQKJNGBBRBMO-UHFFFAOYSA-N110100%active
NQFYAANUFXRFNE-UHFFFAOYSA-N110100%active
QKXWJSXDKHCSDT-LBPRGKRZSA-N110100%active
QKXWJSXDKHCSDT-GFCCVEGCSA-N110100%active
CSFFHTKDUCGKJD-OLZOCXBDSA-N110100%active
CSFFHTKDUCGKJD-STQMWFEESA-N101100%inactive
GJDUQWWYWMTDRL-HNNXBMFYSA-N110100%active
GJDUQWWYWMTDRL-OAHLLOKOSA-N110100%active
HZICFZZGLWKOAR-CVEARBPZSA-N110100%active
HZICFZZGLWKOAR-HOTGVXAUSA-N110100%active
ZMEYPNTUCZBQQN-UHFFFAOYSA-N110100%active
BEWMLXSGKYXKGS-UHFFFAOYSA-N110100%active
ZCRIUCAFIYNTRU-UHFFFAOYSA-N110100%active
NVVCEADQXFTDLA-UHFFFAOYSA-N110100%active
UVDOSWDIUBQDQI-QMMMGPOBSA-N110100%active
UVDOSWDIUBQDQI-MRVPVSSYSA-N110100%active
UJUORBDBVOLWSF-ZJUUUORDSA-N110100%active
UJUORBDBVOLWSF-UWVGGRQHSA-N110100%active
DQGHTEPCNAKPFL-UHFFFAOYSA-N110100%active
UQTTUPZZXWDOQT-UHFFFAOYSA-N110100%active
LPZFCJCYTYLTNK-UHFFFAOYSA-N110100%active
GXSOLYTVGZNXTL-UHFFFAOYSA-N110100%active
DLOOMMVSICCHTJ-UHFFFAOYSA-N110100%active
JSBSVYKRXJJWRJ-UHFFFAOYSA-N101100%inactive
JIHBFKNLUCQAKL-UHFFFAOYSA-N110100%active
AKWFWIHZLMHBGJ-UHFFFAOYSA-N110100%active
MJQGDJQVIHPYTB-UHFFFAOYSA-N110100%active
LPPKYSFULWRWFC-UHFFFAOYSA-N110100%active
ZGXCDVSLCJXLMT-ZDUSSCGKSA-N110100%active
ZGXCDVSLCJXLMT-CYBMUJFWSA-N110100%active
KMZHUPNJAVFPRF-KGLIPLIRSA-N110100%active
KMZHUPNJAVFPRF-KBPBESRZSA-N110100%active
XSSZBQFGRSGRTN-UHFFFAOYSA-N110100%active
URMDJMKUFXNKRG-UHFFFAOYSA-N110100%active
LOVYPHDMDZPQDA-UHFFFAOYSA-N110100%active
YLSPAUGOMPCCCJ-UHFFFAOYSA-N110100%active
XLFNLJYGUOLEJS-SFHVURJKSA-N101100%inactive
FMTZJHHPYOHWNQ-UHFFFAOYSA-N101100%inactive
IEUOMYJAIZIKES-SFQUDFHCSA-N110100%active
SUWNTOBZXIAHKB-CMDGGOBGSA-N110100%active
LPADWFDQODOOMS-DUXPYHPUSA-N101100%inactive
POTINGKLYOETSI-GZTJUZNOSA-N110100%active
DZVIVYUYURSYNH-UHFFFAOYSA-N101100%inactive
MJSXSLBYCSPRHR-UHFFFAOYSA-N101100%inactive
ZVYLAQPDMUKXOT-UHFFFAOYSA-N110100%active
DTQBQXWGJKOUOS-UHFFFAOYSA-N101100%inactive
LNFBAYSBVQBKFR-UHFFFAOYSA-N101100%inactive
SLLRTLCGZRODTB-UHFFFAOYSA-N101100%inactive
WAAWETUDFSIYSD-UHFFFAOYSA-N101100%inactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N101100%inactive
IGRYEDIMNMEBBU-UHFFFAOYSA-N101100%inactive
WHFIWINTCCNYQZ-UHFFFAOYSA-N101100%inactive
UWHWQUTVFLDMPJ-UHFFFAOYSA-N101100%inactive
PAXKGQZKOJPPEG-OLZOCXBDSA-N101100%inactive