P04629 TRKA


Group: TK
Family: Trk
PDB Structure Num: 31
FDA approved drugs from DrugBank: Fostamatinib Imatinib Larotrectinib Regorafenib






structure FDA kinase druginchikeydata countactive numinactive numsame percentagevote label
QMLALHXGVBGFIC-UHFFFAOYSA-N101100%inactive
HSWWFIPPMAFLPH-UHFFFAOYSA-N101100%inactive
NXNQLECPAXXYTR-LCYFTJDESA-N220100%active
KVPNOQAXVUMKFJ-UHFFFAOYSA-N110100%active
UEBUEWAMMXNGMS-LLVKDONJSA-N101100%inactive
BJULBAQIZYUYFI-JTQLQIEISA-N110100%active
SDYJEUJNTJEGGY-HNNXBMFYSA-N110100%active
PGFQSOQKZDCUIL-UHFFFAOYSA-N101100%inactive
SKSUFRGHAZAZHS-UHFFFAOYSA-N110100%active
UEBUEWAMMXNGMS-NSHDSACASA-N110100%active
IZEZSPVHWUPXAH-UHFFFAOYSA-N101100%inactive
MJQVDJSEAMOVCO-UHFFFAOYSA-N110100%active
OOBAQMLMJUYICG-UHFFFAOYSA-N110100%active
XDAYSURCVISUSU-OAHLLOKOSA-N101100%inactive
FXSOVNSBVDXYOV-HNNXBMFYSA-N110100%active
XDAYSURCVISUSU-HNNXBMFYSA-N110100%active
HRMCEFNIUDHQEI-INIZCTEOSA-N110100%active
SDNIEOMSMZTJNX-UHFFFAOYSA-N110100%active
XSRNXUBVNYNCJC-UHFFFAOYSA-N101100%inactive
HIHOEGPXVVKJPP-JTQLQIEISA-N110100%active
JGEBLDKNWBUGRZ-HXUWFJFHSA-N110100%active
WYJRHMPICZARGU-UHFFFAOYSA-N101100%inactive
AEULIVPVIDOLIN-UHFFFAOYSA-N110100%active
GUBJNPWVIUFSTR-UHFFFAOYSA-N110100%active
SPZDCHRXPBSIHM-UHFFFAOYSA-N101100%active
VDKBGBCLPKTOGS-UHFFFAOYSA-N101100%inactive
XYASHXPUZJDWIO-UHFFFAOYSA-N101100%inactive
XLSPYLMTRXPYKY-UHFFFAOYSA-N101100%inactive
CeritinibVERWOWGGCGHDQE-UHFFFAOYSA-N101100%inactive
QKKIWEILHCXECO-UHFFFAOYSA-N110100%active
QHXBWJSQXSYAGG-VIFPVBQESA-N110100%active
DIXMBHMNEHPFCX-MCMMXHMISA-N110100%active
ZKDXRFMOHZVXSG-HNNXBMFYSA-N21150%exclude
LorlatinibIIXWYSCJSQVBQM-LLVKDONJSA-N110100%active
SINWNRPVOPGVAE-UHFFFAOYSA-N21150%exclude
DCLOYUQZPOKYDM-UHFFFAOYSA-N101100%inactive
HTUXRAUCKBVRRI-HXUWFJFHSA-N220100%active
FQGDIYVVDKJSNC-UHFFFAOYSA-N54180%active
OOSFKAZKSXUEGV-UHFFFAOYSA-N220100%active
ZKPYYDAYCYGVLR-UHFFFAOYSA-N220100%active
GKLLTYZVZSJZPP-UHFFFAOYSA-N220100%active
YMPXJQPXFDQSNV-UHFFFAOYSA-N220100%active
AUHGYKJMPIHTCI-UHFFFAOYSA-N21150%exclude
QBTLZXDENPTYFB-UHFFFAOYSA-N21150%exclude
VXBUABPTAFKXED-UHFFFAOYSA-N202100%inactive
JGYGLGXRSWCQPC-UHFFFAOYSA-N220100%active
RFIHHSLMEUBESC-UHFFFAOYSA-N220100%active
YYRGWTNWICCJEY-UHFFFAOYSA-N202100%inactive
AHTITYNYBDULQW-UHFFFAOYSA-N220100%active
BUVASZPZZZNEAY-UHFFFAOYSA-N101100%inactive
MJSHVHLADKXCML-RQNOJGIXSA-N110100%active
ZCHJWXKREFTWSX-UHFFFAOYSA-N101100%inactive
YZOZEZFNWLULHX-UHFFFAOYSA-N101100%inactive
AEBGAQZHEWUQER-UHFFFAOYSA-N101100%inactive
KRMDCWKBEZIMAB-UHFFFAOYSA-N101100%inactive
DADASRPKWOGKCU-FVTQAUBDSA-N110100%active
BNRXMSGHPVYSDK-UHFFFAOYSA-N110100%active
AJDJDSOIQFUPTC-UHFFFAOYSA-N101100%inactive
OXQTXNVWTNDAQF-UHFFFAOYSA-N101100%inactive
ZNMQXOQGTZNCCL-UHFFFAOYSA-N101100%inactive
YUDZZEAZLCNKOZ-UHFFFAOYSA-N110100%active
IXZOFWVKCDIGGX-UHFFFAOYSA-N110100%active
SBPLDFJEHNVMNC-UHFFFAOYSA-N110100%active
BYKSLICDLDTYLA-UHFFFAOYSA-N110100%active
IGJZBYFJOGZJQO-UHFFFAOYSA-N110100%active
WJSPZKYFHWWSDK-UHFFFAOYSA-N110100%active
OGLFUDJJJDTBFS-UHFFFAOYSA-N110100%active
NNDVLAPMFXYAAS-UHFFFAOYSA-N110100%active
NNDVLAPMFXYAAS-FQEVSTJZSA-N101100%inactive
NNDVLAPMFXYAAS-HXUWFJFHSA-N110100%active
RKERQEKFTWWCEY-GOSISDBHSA-N110100%active
AFEWFPBEQADGDP-JOCHJYFZSA-N110100%active
UQKLTKAHTNLXPA-JOCHJYFZSA-N330100%active
QSGGLLCPVRJDDE-JOCHJYFZSA-N330100%active
OHNNRNYUHNGDNO-LSDHHAIUSA-N110100%active
HPNYZOVAOYVLQD-UHFFFAOYSA-N101100%inactive
XVHRKCFLFVJGQU-UHFFFAOYSA-N110100%active
GGFPCEWQWCMOMX-UHFFFAOYSA-N101100%inactive
LTTAHJWMYYUXHI-UHFFFAOYSA-N110100%active
OOCIUHPXHKDTIL-UHFFFAOYSA-N101100%inactive
DJCJLXJLJQLJCL-UHFFFAOYSA-N101100%inactive
SOLRFWOVULTERW-UHFFFAOYSA-N110100%active
JXFUETSWGQSIAJ-UHFFFAOYSA-N110100%active
BDCFBCKBVKPNMH-UHFFFAOYSA-N101100%inactive
MAGVRNDWTTZRHB-UHFFFAOYSA-N110100%active
AEQJHILNCVDPBZ-UHFFFAOYSA-N110100%active
DECBHRUYLCLGGD-UHFFFAOYSA-N101100%inactive
DJYWRQSMWCFDQX-UHFFFAOYSA-N110100%active
SRQQRYTWWRXHKL-UHFFFAOYSA-N110100%active
OSDSLNBKGDENNX-UHFFFAOYSA-N110100%active
NIFOBCJOHDKDIO-UHFFFAOYSA-N110100%active
KYLVMDJXJPCWJF-UHFFFAOYSA-N101100%inactive
OBNFYWGSQNSOJI-UHFFFAOYSA-N101100%inactive
VUNORLWCPMVUBI-UHFFFAOYSA-N101100%inactive
BJSLIJFRTVUWHS-UHFFFAOYSA-N101100%inactive
WGOYYVMNVHOKID-UHFFFAOYSA-N101100%inactive
SZMIXWZBQCALBA-UHFFFAOYSA-N101100%inactive
ZTBYTLSPIBDFPZ-UHFFFAOYSA-N101100%inactive
PRKVTKMWQGQIBO-UHFFFAOYSA-N101100%inactive
PPIXVSWCVIFEMZ-UHFFFAOYSA-N101100%inactive
KQSDCHWZPMZBPP-UHFFFAOYSA-N101100%inactive
HGQXLJWBBLNDTN-UHFFFAOYSA-N101100%inactive
UYXIKIBDQDRVAZ-UHFFFAOYSA-N101100%inactive
CXXCRLLJRGEAJV-UHFFFAOYSA-N101100%inactive
GMTAOJMPNXLKJI-UHFFFAOYSA-N101100%inactive
ZQOTWRRGAAXBIB-UHFFFAOYSA-N110100%active
UXNGTVMJGBIVEX-UHFFFAOYSA-N101100%inactive
UMKXZBLGOSKWKR-UHFFFAOYSA-N101100%inactive
SIQKTWQNQGTCLQ-UHFFFAOYSA-N101100%inactive
XKTJJUVGORXSKR-UHFFFAOYSA-N101100%inactive
RTYGBULZXQMRLX-UHFFFAOYSA-N101100%inactive
SZPJDPHRQQQTIT-UHFFFAOYSA-N101100%inactive
VAIRWATWZQOTMN-UHFFFAOYSA-N101100%inactive
LMDPZAOXFSVSKO-UHFFFAOYSA-N101100%inactive
PQROQALKBIJILZ-UHFFFAOYSA-N101100%inactive
IKUXHAZDRPCANL-UHFFFAOYSA-N101100%inactive
IPMWRJCOSJLTQI-UHFFFAOYSA-N101100%inactive
AXJTYBJJTVPELP-UHFFFAOYSA-N101100%inactive
UOJSYTFKPYHYHF-UHFFFAOYSA-N101100%inactive
QHWYQHKGOYXAON-UHFFFAOYSA-N110100%active
GNNDEPIMDAZHRQ-UHFFFAOYSA-N110100%active
IAZAGXDMMVWYKF-UHFFFAOYSA-N101100%inactive
JDEMVNYMYPJJIM-UHFFFAOYSA-N101100%inactive
SURCGQGDUADKBL-UHFFFAOYSA-N101100%inactive
LarotrectinibNYNZQNWKBKUAII-KBXCAEBGSA-N110100%active
SRKKBPIGHIAVHD-UHFFFAOYSA-N110100%active
CXVBPWYIUWZVJO-UHFFFAOYSA-N110100%active
MMUWXZUTOXDAGI-UHFFFAOYSA-N110100%active
QFQUGVPOOKQVIX-UHFFFAOYSA-N110100%active
YATACVWKJZUENE-VMEOHVCESA-N110100%active
IZHWUQGNICKCJL-OVCLIPMQSA-N110100%active
AGGRVUVLUGVNPX-OVCLIPMQSA-N101100%inactive
QCYYBXWTRITALG-VIZOYTHASA-N110100%active
ZTLMXFXXPNJARJ-UHFFFAOYSA-N110100%active
VLJKEWOJKQIVIX-VAWYXSNFSA-N110100%active
VZAAGSJCIMQODR-UHFFFAOYSA-N110100%active
YVGHJKKTFOXBID-UHFFFAOYSA-N110100%active
DTAWNRUMOCQMSC-LJQANCHMSA-N110100%active
XLFNLJYGUOLEJS-SFHVURJKSA-N110100%active
SQGLEZDWHPDRDX-NZQKXSOJSA-N32166.67%exclude
LBVKEEFIPBQIMD-JTQLQIEISA-N330100%active
IGRYEDIMNMEBBU-UHFFFAOYSA-N101100%inactive
FKQSLMGOZLYGKV-UHFFFAOYSA-N101100%inactive
PUKHKWFFVDCMQS-UHFFFAOYSA-N101100%inactive
URQCQEPGISTGDR-UHFFFAOYSA-N101100%inactive
GBWPNQMIJWWQOK-UHFFFAOYSA-N101100%inactive
DTRNDCUFERMFCI-UHFFFAOYSA-N101100%inactive
IFRLNFINYDTJDH-UHFFFAOYSA-N101100%inactive
KKKVBDXDVWXKRD-UHFFFAOYSA-N101100%inactive
QUJGUPYPJDWQSM-UHFFFAOYSA-N101100%inactive
ALNDBSOOMRQDCM-UHFFFAOYSA-N101100%inactive
YFIBEKZZXUQKCM-UHFFFAOYSA-N101100%inactive
AISDSPKQUIXVOR-UHFFFAOYSA-N110100%active
JVHKMJFKKFFBEZ-UHFFFAOYSA-N110100%active
VWOAWNHKJWXMQE-UHFFFAOYSA-N101100%inactive
WZGCSCUTQNHMDL-UHFFFAOYSA-N101100%inactive
RYDVHEGEODXHRQ-UHFFFAOYSA-N101100%inactive
HTRIQCMSXMSDKF-UHFFFAOYSA-N101100%inactive
LHKSZDXILCOKIZ-UHFFFAOYSA-N101100%inactive
HQWSGBYYANMPKM-UHFFFAOYSA-N101100%inactive
WYQSOSKRGKZWFS-UHFFFAOYSA-N101100%inactive
MFDOFMCHLFWXLY-UHFFFAOYSA-N101100%inactive
HMYJNQKCQFDTEW-UHFFFAOYSA-N101100%inactive
BTGLGOLMMONDLB-UHFFFAOYSA-N101100%inactive
MGYZMBWNGIKJEE-UHFFFAOYSA-N110100%active
OYFHGYBLCJITBK-UHFFFAOYSA-N101100%inactive
UXFSFDLEUWWWLP-UHFFFAOYSA-N101100%inactive
WRPKJOAKDSVTBN-UHFFFAOYSA-N101100%inactive
RKGGNRKEAHCEBE-UHFFFAOYSA-N101100%inactive
PUULXMCIENDJKJ-UHFFFAOYSA-N101100%inactive
RFZKWTPDLFQYIS-UHFFFAOYSA-N101100%inactive
YJDGFZVIIUFVIV-UHFFFAOYSA-N101100%inactive
PKAMBYZNJPJUFT-UHFFFAOYSA-N101100%inactive
ULDMDFPXNRGXSE-UHFFFAOYSA-N110100%active
COXZOGYEXZWLMM-UHFFFAOYSA-N101100%inactive
VERHZRWOVSXMOW-UHFFFAOYSA-N110100%active
JWILUIVAYLRFIY-UHFFFAOYSA-N110100%active
KOZFSFOOLUUIGY-SOLYNIJKSA-N220100%active
MDAFGVXLBFQEJH-XCFOVOSNSA-N110100%active
CVXZWDPKRAIHOI-SVQPHZEZSA-N110100%active
UFKSWYKDQZBJTH-UHFFFAOYSA-N101100%inactive
HXGMCPSJILOUIU-IHMJZKOGSA-N110100%active
HXGMCPSJILOUIU-LROUJFHJSA-N220100%active
NMMGUHANGUWNBN-VHEIIQRDSA-N110100%active
BIJVEGOYPDBWSR-CXAHNHKCSA-N110100%active
ONSKSKMJNHEONW-WINIVTDRSA-N110100%active
ONSKSKMJNHEONW-XHCCPWGMSA-N110100%active
KOZFSFOOLUUIGY-BLIZRMSTSA-N220100%active
NTMHCRKKNMVCAH-UHFFFAOYSA-N110100%active
ZZRZYNUVVRVWRW-UHFFFAOYSA-N110100%active
QKNIGHXAMOUFPM-UHFFFAOYSA-N110100%active
UWEPEBZEGMXIMW-UHFFFAOYSA-N110100%active
MVNXGVRGJAIDMD-UHFFFAOYSA-N101100%inactive
HYEDJICMYMBSHW-UHFFFAOYSA-N110100%active
VKPWSFHSZDMYGW-UHFFFAOYSA-N110100%active
YSOVXPTZPIBWGX-UHFFFAOYSA-N110100%active
HEEKPDWNVFGASY-SNVBAGLBSA-N110100%active
AARWOJHWGOYIRM-UHFFFAOYSA-N110100%active
LHKRNWZSFJYSNE-UHFFFAOYSA-N110100%active
HEEKPDWNVFGASY-JTQLQIEISA-N110100%active
DLMDRALHZSWJSF-UHFFFAOYSA-N110100%active
GQFFWPAHFXPYSA-UHFFFAOYSA-N110100%active
SVAHIJWZHJDMBM-UHFFFAOYSA-N110100%active
ZAQBXBCUJGIFKY-UHFFFAOYSA-N110100%active
MZLDGXSGVBFEPD-UHFFFAOYSA-N110100%active
OYVOITSEETVYOR-UHFFFAOYSA-N110100%active
OJNYWHSZTYNGPE-UHFFFAOYSA-N110100%active
NMUIYMCYQWYFCA-UHFFFAOYSA-N101100%inactive
HEEKPDWNVFGASY-UHFFFAOYSA-N110100%active
HEBJWJMMXHCUJW-UHFFFAOYSA-N110100%active
HHKGVQGXRGQBBA-UHFFFAOYSA-N101100%inactive
GMVQPWCWWLPOQT-FQEVSTJZSA-N110100%active
XKFTZKGMDDZMJI-HSZRJFAPSA-N110100%active
ABMSAGZBJYEZGT-UHFFFAOYSA-N110100%active
WENCWJUIDFEPSK-UHFFFAOYSA-N110100%active
NBGYLHIDCLVBHE-UHFFFAOYSA-N110100%active
NNBUSHQYRIXNJY-XOBRGWDASA-N110100%active
FNCGOKWVESVXSF-VLIAUNLRSA-N110100%active
JVJZHQKVZJRSQR-QKKBWIMNSA-N110100%active
PFEHGXFVDGRZKZ-OSPHWJPCSA-N110100%active
HLFAQOKXVIJWBD-YJYMSZOUSA-N110100%active
PFEHGXFVDGRZKZ-XDHUDOTRSA-N110100%active
JVJZHQKVZJRSQR-SZNDQCEHSA-N110100%active
NNBUSHQYRIXNJY-VLIAUNLRSA-N110100%active
FNCGOKWVESVXSF-XOBRGWDASA-N110100%active
HLFAQOKXVIJWBD-DJJJIMSYSA-N110100%active
ZATWYMPHUYHZKA-LLVKDONJSA-N220100%active
QJVHIMLGONEYEE-UHFFFAOYSA-N110100%active
UZWKONVGWZDEMU-UHFFFAOYSA-N110100%active
DBEUDOPZCCISRU-UHFFFAOYSA-N110100%active
OKQYVMVRBRSVES-UHFFFAOYSA-N110100%active
ZATWYMPHUYHZKA-UHFFFAOYSA-N110100%active
FOQGKYFZJPXSNG-UHFFFAOYSA-N101100%inactive
UKZRGBUTBINTPD-LOSJGSFVSA-N202100%inactive
PNMQDIXULZYDDT-UHFFFAOYSA-N202100%inactive
YGLAORIVGOGYSS-UHFFFAOYSA-N101100%inactive
WWUXHXQJFWXACS-UHFFFAOYSA-N101100%inactive
OUBLXGAHJPBMHW-UHFFFAOYSA-N101100%inactive
NWEIOMWQAHZBEE-UHFFFAOYSA-N101100%inactive
BQCBWCAJXUXWIA-UHFFFAOYSA-N101100%inactive
OWLAKERMHYDWTB-UHFFFAOYSA-N101100%inactive
FGNQVZZMORDWIZ-UHFFFAOYSA-N101100%inactive
GIAVVFIPFBOBRR-UHFFFAOYSA-N101100%inactive
QPVNTDBWWRFMIC-UHFFFAOYSA-N101100%inactive
QUYGYUVUHYMMRW-UHFFFAOYSA-N101100%inactive
HRDSLRKPXDHOAX-UHFFFAOYSA-N101100%inactive
XOWDXZZFGKMQIB-UHFFFAOYSA-N101100%inactive
ARYVAQSYRLZVQD-UHFFFAOYSA-N101100%inactive
WAAWETUDFSIYSD-UHFFFAOYSA-N101100%inactive
ZEHBZHZMQSHZFI-UHFFFAOYSA-N101100%inactive
IUZVIJYTCSDYGR-UHFFFAOYSA-N101100%inactive
SZVCJSVITVKTQV-UHFFFAOYSA-N101100%inactive
HDJKZMBKHFPSSU-UHFFFAOYSA-N101100%inactive
NFYWVJCAMOJHHV-UHFFFAOYSA-N101100%inactive
BYHRBRFVUCUWQO-UHFFFAOYSA-N101100%inactive
MVWVWWBAONWJOC-UHFFFAOYSA-N101100%inactive
WALGXADGJIZYNY-UHFFFAOYSA-N101100%inactive
WDUHSVJZBUZHNP-UHFFFAOYSA-N101100%inactive
FOGGTLYHDTZVPS-UHFFFAOYSA-N101100%inactive
ZEYJXRCHEFTSTA-UHFFFAOYSA-N101100%inactive
LEZPQBWEYFVLLL-UHFFFAOYSA-N101100%inactive
MKYBMEVSJFNENA-UHFFFAOYSA-N101100%inactive
ROVFNLCGTHSKOF-UHFFFAOYSA-N101100%inactive
GPWYEGZCLUSIDX-UHFFFAOYSA-N101100%inactive
SNSKMGFZGTWQSI-UHFFFAOYSA-N101100%inactive
MFEXYTURXUZOID-UHFFFAOYSA-N101100%inactive
IYBYMTCQQMFOHB-AATRIKPKSA-N101100%inactive
MDWXVGCLSBQVMP-UHFFFAOYSA-N101100%inactive
FMTZJHHPYOHWNQ-UHFFFAOYSA-N101100%inactive
WHFIWINTCCNYQZ-UHFFFAOYSA-N101100%inactive
XKXRQJGEXCKDGJ-UHFFFAOYSA-N101100%inactive
TUNDWEPBBZFASQ-UHFFFAOYSA-N101100%inactive
WDNYTEIRGJADIJ-UHFFFAOYSA-N101100%inactive
AJJJGWBGCBQBHY-UHFFFAOYSA-N101100%inactive
GVRQPZHEXGIECW-UHFFFAOYSA-N101100%inactive
GXXLIFVPMIUTRC-UHFFFAOYSA-N101100%inactive
IETYBEPYBOFTIR-UHFFFAOYSA-N101100%inactive
ACIJUAXTIRFXDI-UHFFFAOYSA-N101100%inactive
XESHALHZSKFLSE-UHFFFAOYSA-N101100%inactive
SCMLRESZJCKCTC-SVQPHZEZSA-N101100%inactive
SIHPNVHZKXZMMW-HPXOIRBESA-N101100%inactive
FPXKTABMRKRDJN-HPXOIRBESA-N101100%inactive
CMAAJKFJPMUHEN-GWAZHQGNSA-N101100%inactive
XIKCRRWSJXYZMA-HPXOIRBESA-N101100%inactive
MLIFNJABMANKEU-UHFFFAOYSA-N101100%inactive
CXVCCFWINYQPRS-UHFFFAOYSA-N101100%inactive
PFFVLVCIEPYEFP-UHFFFAOYSA-N101100%inactive
RAOJISQDGOOXTK-UHFFFAOYSA-N101100%inactive
NHDDTLMPCVOXFH-UHFFFAOYSA-N101100%inactive